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Naloxone is an antagonist of Opioid receptor. Naloxone alleviates opioid-overdose-induced respiratory depression. Naloxone may cause pulmonary edema and cardiac arrhythmias [1]. Uses: Scientific research. Group: Signaling pathways. CAS No. 465-65-6. Pack Sizes: 10 mg; 25 mg; 50 mg; 100 mg; 200 mg. Product ID: HY-17417A.
Naloxone benzoylhydrazone
Naloxone benzoylhydrazone. Group: Biochemicals. Grades: Purified. CAS No. 119630-94-3. Pack Sizes: 10mg, 50mg. US Biological Life Sciences.
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Naloxone benzoylhydrazone
Naloxone benzoylhydrazone (NalBzoH) is a mixed agonist/antagonist. Naloxone benzoylhydrazone is a prototypic κ3-opioid receptor agonist, and a partial agonist at the cloned μ and δ opioid receptors , and an antagonist at opioid-like NOP receptors. Naloxone benzoylhydrazone has potently analgesia effect [1] [2] [3]. Uses: Scientific research. Group: Signaling pathways. Alternative Names: NalBzoH. CAS No. 119630-94-3. Pack Sizes: 1 mg. Product ID: HY-107743.
Naloxone EP Impurity B
Naloxone EP Impurity B. Uses: For analytical and research use. Group: Impurity standards. CAS No. 1352085-46-1. Molecular Formula: C22H25NO4. Mole Weight: 367.44. Catalog: APB1352085461.
Naloxone EP Impurity C
Naloxone EP Impurity C. Uses: For analytical and research use. Group: Impurity standards. CAS No. 2139253-68-0. Molecular Formula: C19H21NO5. Mole Weight: 343.38. Catalog: APB2139253680.
Naloxone EP Impurity F
Naloxone EP Impurity F. Uses: For analytical and research use. Group: Impurity standards. CAS No. 2139253-69-1. Molecular Formula: C19H21NO5. Mole Weight: 343.38. Catalog: APB2139253691.
Naloxone EP Impurity G
Naloxone EP Impurity G. Uses: For analytical and research use. Group: Impurity standards. CAS No. 70866-64-7. Molecular Formula: C20H23NO4. Mole Weight: 341.41. Catalog: APB70866647.
Naloxone hydrochloride
Naloxone hydrochloride. Group: Biochemicals. Grades: Purified. CAS No. 357-08-4. Pack Sizes: 100mg. US Biological Life Sciences.
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Naloxone hydrochloride
Naloxone hydrochloride is an antagonist of Opioid receptor. Naloxone hydrochloride alleviates opioid-overdose-induced respiratory depression. Naloxone hydrochloride may cause pulmonary edema and cardiac arrhythmias [1]. Uses: Scientific research. Group: Signaling pathways. CAS No. 357-08-4. Pack Sizes: 100 mg; 500 mg. Product ID: HY-17417.
Naloxone Impurity 8
Naloxone Impurity 8. Uses: For analytical and research use. Group: Impurity standards. Molecular Formula: C31H48N2O12. Mole Weight: 640.73. Catalog: APB08711.
Naloxone methiodide
Naloxone methiodide is a peripherally restricted, nonselective, and competitive opioid receptor antagonist. Naloxone methiodide does not penetrate the blood-brain barrier [1] [2]. Uses: Scientific research. Group: Signaling pathways. CAS No. 93302-47-7. Pack Sizes: 1 mg. Product ID: HY-137279.
10-Keto Naloxone
10-Keto Naloxone. Uses: For analytical and research use. Group: Impurity standards. CAS No. 294175-43-2. Molecular Formula: C19H19NO5. Mole Weight: 341.36. Catalog: APB294175432.
14-Chloro Naloxone
14-Chloro Naloxone. Uses: For analytical and research use. Group: Impurity standards. Molecular Formula: C19H20ClNO3. Mole Weight: 345.82. Catalog: APB08710.
2,2-Bisnaloxone
2,2-Bisnaloxone is an impurity of Naloxone (N285000), a specific opioid antagonist and narcotic antagonist. Group: Biochemicals. Grades: Highly Purified. CAS No. 211738-08-8. Pack Sizes: 5mg, 50mg. Molecular Formula: C38H40N2O8. US Biological Life Sciences.
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(10α, 8 β)-Dihydroxy Naltrexone
(10α, 8 β)-Dihydroxy Naltrexone is a derivative of Naltrexone (N285750), a nonselective opioid receptor antagonist; congener of Naloxone. Group: Biochemicals. Grades: Highly Purified. Pack Sizes: 1mg, 2.5mg. Molecular Formula: C20H23NO6, Molecular Weight: 373.4. US Biological Life Sciences.
Worldwide
10α-Hydroxy Naltrexone
10α-Hydroxy Naltrexone is a derivative of Naltrexone (N285750), a nonselective opioid receptor antagonist; congener of Naloxone. Group: Biochemicals. Grades: Highly Purified. Pack Sizes: 1mg, 2.5mg. Molecular Formula: C20H23NO5, Molecular Weight: 357.4. US Biological Life Sciences.
Worldwide
(10 β, 8 β)-Dihydroxy Naltrexone
(10 β, 8 β)-Dihydroxy Naltrexone is a derivative of Naltrexone (N285750), a nonselective opioid receptor antagonist; congener of Naloxone. Group: Biochemicals. Grades: Highly Purified. Pack Sizes: 1mg, 2.5mg. Molecular Formula: C20H23NO6, Molecular Weight: 373.4. US Biological Life Sciences.
Worldwide
10 β-Hydroxy Naltrexone
10 β-Hydroxy Naltrexone is a derivative of Naltrexone (N285750), a nonselective opioid receptor antagonist; congener of Naloxone. Group: Biochemicals. Grades: Highly Purified. Pack Sizes: 1mg, 2.5mg. Molecular Formula: C20H23NO5, Molecular Weight: 357.4. US Biological Life Sciences.
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10-Hydroxy Norhydrocodone
10-Hydroxy Norhydrocodone is an iintermediate in the synthesis of Naloxone (HCl salt, N285000) related compounds as opioid antagonist and narcotic antagonist. Group: Biochemicals. Grades: Highly Purified. Pack Sizes: 50mg, 100mg. Molecular Formula: C17H19NO4, Molecular Weight: 301.339999999999. US Biological Life Sciences.
Worldwide
14-Hydroxy Norcodeinone
14-Hydroxy Norcodeinone is an inertermediate in the synthesis of N-Allyldi hydro-8, 10, 14-tri hydroxynormorphinone (A549610), an impurity of Naloxone (HCl salt, N285000) which is a specific opioid antagonist and narcotic antagonist. Group: Biochemicals. Grades: Highly Purified. CAS No. 2302-68-3. Pack Sizes: 1mg, 2.5mg. Molecular Formula: C17H17NO4, Molecular Weight: 299.32. US Biological Life Sciences.
Worldwide
1-Chloro Naltrexone
1-Chloro Naltrexone is a derivative of Naloxone, which is used to treat alcohol dependence and prevent relapse of opioid dependence. Molecular formula: C20H22ClNO4. Mole weight: 375.85.
1-Chloro Naltrexone
1-Chloro Naltrexone is a derivative of Naltrexone (N285750), a nonselective opioid receptor antagonist; congener of Naloxone. Group: Biochemicals. Grades: Highly Purified. Pack Sizes: 1mg, 2.5mg. Molecular Formula: C20H22ClNO4, Molecular Weight: 375.85. US Biological Life Sciences.
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2-Chloro-10-hydroxynaltrexone
2-Chloro-10-hydroxynaltrexone is a naltrexone degradant from REVIA tablets. Also, it is derived from the parent compound Naltrexone Hydrochloride (N285750), a non-selective opioid receptor antagonist; congener of Naloxone. Group: Biochemicals. Grades: Highly Purified. CAS No. 619331-76-9. Pack Sizes: 1mg. Molecular Formula: C20H22ClNO5, Molecular Weight: 391.85. US Biological Life Sciences.
Worldwide
2-Chloro Naltrexone
2-Chloro Naltrexone is a derivative of Naltrexone (N285750), a nonselective opioid receptor antagonist; congener of Naloxone. Group: Biochemicals. Grades: Highly Purified. Pack Sizes: 1mg, 2.5mg. Molecular Formula: C20H22ClNO4, Molecular Weight: 375.85. US Biological Life Sciences.
(4R,4aS,12bS)-3-allyl-7-propoxy-2,3,4,4a,5,7a-hexahydro-1H-4,12-methanobenzofuro[3,2-e]isoquinoline-4a,9-diol is a synthetic analog of Naloxone, which is a medication used to reverse the effects of opioids. Molecular formula: C22H27NO4. Mole weight: 369.45.
(5α)-4,5-Epoxy-14-hydroxy-2-iodo-3-methoxy-17-(2-propen-1-yl)-morphinan-6-one Cyclic 1,2-Ethanediyl Acetal is a synthetic analog of Naloxone, which is a medication used to reverse the effects of opioids. Molecular formula: C22H26INO5. Mole weight: 511.35.
CCK (27-33) (non-sulfated)
Cholecystokinin (CCK) is a neuropeptide and gut hormone that regulates pancreatic enzyme secretion and gastrointestinal motility, and acts as a satiety signal. CCK (27-33) is a C-terminal fragment of CCK. Non-sulfated CCK (27-33) inhibits binding of [3H]naloxone in rat cerebellum membranes with IC50 of 4 μM and inhibits electrically-stimulated contraction of isolated guinea pig ileum with IC50 of 17 μM. Synonyms: Cholecystokinin (27-33) (non-sulfated). Grades: ≥95%. CAS No. 47910-79-2. Molecular formula: C45H57N9O10S2. Mole weight: 948.12.
ICI 174864
ICI 174864 is a highly selective, potent δ-receptor antagonist. ICI 174864 is equipotent with naloxone and can not reverse the effect of the μ-agonist [D-Ala2, MePhe4, Gly-Ol5]enkephalin or the κ-agonist-tifluadom [1]. Uses: Scientific research. Group: Peptides. CAS No. 89352-67-0. Pack Sizes: 1 mg. Product ID: HY-101230.
morphine 6-dehydrogenase
Also acts on some other alkaloids, including codeine, normorphine and ethylmorphine, but only very slowly on 7,8-saturated derivatives such as dihydromorphine and dihydrocodeine. In the reverse direction, also reduces naloxone to the 6α-hydroxy analogue. Activated by 2-mercaptoethanol. Group: Enzymes. Synonyms: naloxone reductase; reductase, naloxone. Enzyme Commission Number: EC 1.1.1.218. CAS No. 97002-71-6. Storage: Store it at +4 ?C for short term. For long term storage, store it at -20 ?C?-80 ?C. Form: Liquid or lyophilized powder. EXWM-0123; morphine 6-dehydrogenase; EC 1.1.1.218; 97002-71-6; naloxone reductase; reductase, naloxone. Cat No: EXWM-0123.
Nonselective opioid receptor antagonist; congener of naloxone. Group: Biochemicals. Alternative Names: (5a)-17-(Cyclopropyl-methyl)-4,5-epoxy-3,14-dihydroxymorphinan-6-one-d3. Grades: Highly Purified. Pack Sizes: 1mg. US Biological Life Sciences.
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Naltrexone Hydrochloride
Nonselective opioid receptor antagonist; congener of Naloxone. Group: Biochemicals. Alternative Names: (5α)-17-(Cyclopropyl-methyl-d3)-4,5-epoxy-3,14-dihydroxymorphinan-6-one Hydrochloride; Antaxone; Depade; EN 1639A; NIH 8503; Nalorex; Trexan. Grades: Highly Purified. CAS No. 16676-29-2. Pack Sizes: 250mg. US Biological Life Sciences.
Worldwide
PD-117302
PD-117302, a new nonpeptide opioid compound, is a selective kappa-opioid agonist. It has been evaluated in vivo for antinociceptive activity and other effects characteristic of kappa-receptor activation. It also causes naloxone-reversible locomotor impairment and diuresis. It is used as an Anticonvulsants, an Anti-Arrhythmia agent, a Central Nervous System agent and a Cardiovascular agent. Uses: Pd-117302 is used as an anticonvulsants, an anti-arrhythmia agent, a central nervous system agent and a cardiovascular agent. Synonyms: PD117302; PD-117302; PD 117302; Trans-N-Methyl-N-(2-(1-pyrrolidinyl)cyclohexyl-)benzo-(b)-thiophene-4-acetamide;Benzo(b)thiophene-4-acetamide, N-methyl-N-(2-(1-pyrrolidinyl)cyclohexyl)-, trans-(+-)-;2-(1-Benzothiophen-4-yl)-N-methyl-N-[(1R,2R)-2-pyrrolidin-1-ylcyclohexyl]acetamide;PD117302. Grades: >98%. CAS No. 111728-01-9. Molecular formula: C21H28N2OS. Mole weight: 356.52.
Naloxonazine dihydrochloride
Naloxonazine dihydrochloride. Group: Biochemicals. Grades: Purified. CAS No. 880759-65-9. Pack Sizes: 10mg, 50mg. US Biological Life Sciences.
Worldwide
Naloxonazine dihydrochloride
Naloxonazine dihydrochloride is a potent and selective antagonist for μ1 opioid receptors. Studies show that pretreatment with naloxonazine significantly attenuated the acute METH-induced increase in locomotor activity and phosphor-Thr75 DARPP-32 levels. Synonyms: Bis-[5-α-4,5-Epoxy-3,14-dihydroxy-17-(2-propenyl)-morphinan-6-ylidene] hydrazine dihydrochloride; Naloxonazine Dihydrochloride; Naloxonazine 2HCl. Grades: ≥98% by HPLC. CAS No. 880759-65-9. Molecular formula: C38H42N4O6.2HCl. Mole weight: 723.69.
Naloxonazine dihydrochloride
Naloxonazine dihydrochloride is a specific μ-opioid receptor antagonist with an IC 50 of 5.4 nM. Naloxonazine dihydrochloride also shows anti-leishmanial activity [1] [2] [3]. Uses: Scientific research. Group: Signaling pathways. CAS No. 880759-65-9. Pack Sizes: 5 mg. Product ID: HY-101011.
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