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| Product | Description | |
|---|---|---|
| Endomorphin 1 | Endomorphin 1, a high affinity, highly selective agonist of the μ-opioid receptor ( K i : 1.11 nM), displays reasonable affinities for kappa 3 binding sites, with K i value between 20 and 30 nM. Endomorphin 1 has antinociceptive properties [1] [2] [4]. Uses: Scientific research. Group: Peptides. CAS No. 189388-22-5. Pack Sizes: 10 mM * 1 mL; 5 mg; 10 mg; 25 mg. Product ID: HY-P0185. |  |
| Endomorphin 1 | Endomorphin 1 is a high affinity (Ki = 360 pM) and highly selective agonist of theμ-opioid receptor with 4000- and 15000-fold preference over δ and κ respectively and displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM. Uses: Analgesics, opioid. Synonyms: L-tyrosyl-L-prolyl-L-tryptophyl-L-phenylalaninamide. CAS No. 189388-22-5. Molecular formula: C34H38N6O5. Mole weight: 610.7. |  |
| Endomorphin 1 acetate | Endomorphin 1 acetate, a high affinity, highly selective agonist of the μ-opioid receptor ( K i : 1.11 nM), displays reasonable affinities for kappa 3 binding sites, with K i value between 20 and 30 nM. Endomorphin 1 acetate has antinociceptive properties [1] [2] [4]. Uses: Scientific research. Group: Peptides. CAS No. 1276123-71-7. Pack Sizes: 5 mg; 10 mg; 25 mg. Product ID: HY-P0185A. | |
| Endomorphin 1 trifluoroacetate salt | Endomorphin 1, an endogenous neuropeptide, is found in the brain and, to a lesser extent, in the spinal cord. It is an agonist of μ-opioid receptor (Ki = 0.36 nM) that has analgesic, positive reinforcing, and gastrointestinal properties, which is selective for μ- over δ- and κ-opioid receptors (Ki = 1,506 and 5,428 nM, respectively). Synonyms: L-tyrosyl-L-prolyl-L-tryptophyl-L-phenylalaninamide, trifluoroacetate salt. Grade: ≥95%. Molecular formula: C34H38N6O5·xCF3COOH. Mole weight: 610.70. | |
| N-terminally acetylated Endomorphin-1 | N-terminally acetylated Endomorphin-1 is a modified Endomorphin-1. Synonyms: Ac-L-Tyr-L-Pro-L-Trp-L-Phe-CONH2; H-Tyr(Ac)-Pro-Trp-Phe-NH2; Ac-LYLPLWLF-NH2; O4-acetyl-L-tyrosyl-L-prolyl-L-tryptophyl-L-phenylalaninamide. Grade: ≥95%. Molecular formula: C36H40N6O6. Mole weight: 652.74. | |
| N-terminally acetylated Endomorphin-1 acetate | N-terminally acetylated Endomorphin-1 is a modified Endomorphin-1. Molecular formula: C38H44N6O8. Mole weight: 712.79. | |
| BMS 986122 | BMS 986122 is a positive allosteric modulator of the μ-Opioid receptor. It significantly increases the inhibition of forskolin-stimulated adenylyl cyclase activity produced by an EC10 (30 pM) concentration of endomorphin-I in CHO-μ cells. BMS 986122 potentiates endomorphin 1-induced inhibition of forskolin-stimulated adenylyl cyclase activity in CHO cells expressing human recombinant μ-opioid receptors with EC50 of 8.9 μM. It also enhances [35S]GTPγ binding stimulated by the μ-opioid agonist DAMGO by 7- and 4.5-fold in C6μ glioma cell membranes. Synonyms: BMS-986122; BMS986122; 2-(3-bromo-4-methoxyphenyl)-3-[(4-chlorophenyl)sulfonyl]-thiazolidine. Grade: ≥98%. CAS No. 313669-88-4. Molecular formula: C16H15BrClNO3S2. Mole weight: 448.8. | |
| BMS 986188 | BMS 986188 is a novel potent and selective positive allosteric modulator of the delta-opioid receptor. It is selective for δ- over μ-opioid receptors with EC50 of 10 μM in the presence of leu-enkephalin and the μ-opioid receptor agonist endomorphin 1, respectively. Synonyms: MS-986188; BMS 986188. Grade: ≥98%. CAS No. 1776115-10-6. Molecular formula: C30H31BrO4. Mole weight: 535.5. | |
| Endomorphin 2 | Endomorphin 2, an andogenous peptide, has high affinity and specificity for the μ-opioid receptor and displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM. Uses: Analgesics, opioid. Synonyms: H-Tyr-Pro-Phe-Phe-NH2; L-tyrosyl-L-prolyl-L-phenylalanyl-L-phenylalaninamide; (2S)-1-[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]-N-[(2S)-1-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]pyrrolidine-2-carboxamide. Grade: >95%. CAS No. 141801-26-5. Molecular formula: C32H37N5O5. Mole weight: 571.7. | |
| Endomorphin 2 TFA | Endomorphin 2 TFA, a high affinity, highly selective agonist of the μ-opioid receptor , displays reasonable affinities for kappa 3 binding sites, with K i value between 20 and 30 nM [1]. Uses: Scientific research. Group: Peptides. CAS No. 1276124-00-5. Pack Sizes: 10 mM * 1 mL; 5 mg; 10 mg; 25 mg. Product ID: HY-P0186A. | |
| Endomorphin 2 TFA | Endomorphin 2 TFA is a high affinity, highly selective agonist of the μ-opioid receptor. It displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM. Synonyms: Endomorphin 2 (TFA); Endomorphin-2 Trifluoroacetate; L-tyrosyl-L-prolyl-L-phenylalanyl-L-phenylalaninamide,trifluoroacetatesalt. Grade: 99%. CAS No. 1276124-00-5. Molecular formula: C34H38F3N5O7. Mole weight: 685.69. | |
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