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Product | Description | |
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Abl Cytosolic Substrate Quick inquiry Where to buy Suppliers range | Abl Cytosolic Substrate is a substrate for Abelson tyrosine kinase (Abl). Synonyms: L-Lysine, L-α-glutamyl-L-alanyl-L-isoleucyl-L-tyrosyl-L-alanyl-L-alanyl-L-prolyl-L-phenylalanyl-L-alanyl-L-lysyl-L-lysyl-; L-Lysine, N2-[N2-[N2-[N-[N-[1-[N-[N-[N-[N-(N-L-α-glutamyl-L-alanyl)-L-isoleucyl]-L-tyrosyl]-L-alanyl]-L-alanyl]-L-prolyl]-L-phenylalanyl]-L-alanyl]-L-lysyl]-L-lysyl]-; L-α-Glutamyl-L-alanyl-L-isoleucyl-L-tyrosyl-L-alanyl-L-alanyl-L-prolyl-L-phenylalanyl-L-alanyl-L-lysyl-L-lysyl-L-lysine; Glu-Ala-Ile-Tyr-Ala-Ala-Pro-Phe-Ala-Lys-Lys-Lys. Grades: ≥95%. CAS No. 168202-46-8. Molecular formula: C64H101N15O16. Mole weight: 1336.58. | |
Abl Cytosolic Substrate Quick inquiry Where to buy Suppliers range | Abl Cytosolic Substrate is a substrate for Abelson tyrosine kinase (Abl ). Abl Protein Tyrosine Kinase (AbI) is a truncated form of the v-AbI Protein Tyrosine Kinase, a partner in the Gag-Abl fusion protein of the Abelson murine leukemia virus. Uses: Peptide Inhibitors. CAS No. 168202-46-8. Product ID: R1142. | |
Abl Cytosolic Substrate acetate Quick inquiry Where to buy Suppliers range | Abl Cytosolic Substrate acetate is a substrate for Abelson tyrosine kinase (Abl). Synonyms: Glu-Ala-Ile-Tyr-Ala-Ala-Pro-Phe-Ala-Lys-Lys-Lys acetate salt; L-α-Glutamyl-L-alanyl-L-isoleucyl-L-tyrosyl-L-alanyl-L-alanyl-L-prolyl-L-phenylalanyl-L-alanyl-L-lysyl-L-lysyl-L-Lysine acetate salt. Grades: ≥95%. CAS No. 2918768-10-0. Molecular formula: C64H101N15O16.C2H4O2. Mole weight: 1396.63. | |
10β-Hydroperoxy Norethindrone Acetate Quick inquiry Where to buy Suppliers range | 10β-Hydroperoxy Norethindrone Acetate is a derivative of Norethindrone, which is an oral contraceptive involved in the inhibition of cytosolic sulfotransferases. Synonyms: 10-Hydroperoxy-17-hydroxy-19-nor-17α-pregn-4-en-20-yn-3-one 17-Acetate; Norethindrone Impurity 4; 19-Nor-17α-pregn-4-en-20-yn-3-one, 10-hydroperoxy-17-hydroxy-, 17-acetate; Norethindrone Acetate Impurity 15. CAS No. 13236-11-8. Molecular formula: C22H28O5. Mole weight: 372.45. | |
10-beta Hydroxy Norethindrone Quick inquiry Where to buy Suppliers range | An impurity of Norethindrone, which is an oral contraceptive involved in the inhibition of cytosolic sulfotransferases. Synonyms: 10β-Hydroxy Norethindrone; (17α)-10,17-Dihydroxy-19-norpregn-4-en-20-yn-3-one; 10,17-Dihydroxy-19-nor-17α-pregn-4-en-20-yn-3-one. Grades: > 95%. CAS No. 1236-00-6. Molecular formula: C20H26O3. Mole weight: 314.43. | |
16β-Hydroxy-17-epi-norethisterone Quick inquiry Where to buy Suppliers range | 16β-Hydroxy-17-epi-norethisterone is an impurity of Norethindrone, which is an oral contraceptive involved in the inhibition of cytosolic sulfotransferases. Synonyms: 16β,17-Dihydroxy-19-norpregn-4-en-20-yn-3-one; 16β-Hydroxy-18-methyllevonorgestrel; (8R,9S,10R,13S,14S,16R,17S)-17-ethynyl-16,17-dihydroxy-13-methyl-1,2,6,7,8,9,10,11,12,14,15,16-dodecahydrocyclopenta[a]phenanthren-3-one. Molecular formula: C20H26O3. Mole weight: 314.42. | |
(17α)-17-Hydroxy-19-norpregn-5-en-20-yn-3-one Cyclic 1,2-Ethanediyl Acetal Quick inquiry Where to buy Suppliers range | (17α)-17-Hydroxy-19-norpregn-5-en-20-yn-3-one Cyclic 1,2-Ethanediyl Acetal is an impurity of Norethindrone, which is an oral contraceptive involved in the inhibition of cytosolic sulfotransferases. Synonyms: Spiro[3H-cyclopenta[a]phenanthrene-3,2'-[1,3]dioxolane] 19-Norpregn-5-en-20-yn-3-one deriv.; Spiro[3H-cyclopenta[a]phenanthrene-3,2'-[1,3]dioxolan]-17-ol, 17-ethynyl-1,2,4,7,8,9,10,11,12,13,14,15,16,17-tetradecahydro-13-methyl-, (8R,9S,10R,13S,14S,17R)-. CAS No. 22170-58-7. Molecular formula: C22H30O3. Mole weight: 342.47. | |
(17α)-19-Norpregn-5-en-20-yne-3,17-diol Quick inquiry Where to buy Suppliers range | (17α)-19-Norpregn-5-en-20-yne-3,17-diol is an intermediate in the preparation of Norethindrone, which is an oral contraceptive involved in the inhibition of cytosolic sulfotransferases. Synonyms: Norethindrone Impurity 36; (8R,9S,10R,13S,14S,17R)-17-ethynyl-13-methyl-2,3,4,7,8,9,10,11,12,13,14,15,16,17-tetradecahydro-1H-cyclopenta[a]phenanthrene-3,17-diol; Estr-5-ene-3,17-diol, 17-ethynyl-, (17β)-. Grades: ≥95%. CAS No. 1492-41-7. Molecular formula: C20H28O2. Mole weight: 300.43. | |
17α-Cyanomethyl-19-nortestosterone Quick inquiry Where to buy Suppliers range | 17α-Cyanomethyl-19-nortestosterone is a metabolite of Norethindrone, which is an oral contraceptive involved in the inhibition of cytosolic sulfotransferases. Synonyms: STS 384; STS 528; 17α-Cyanomethyl-17β-hydroxyestr-4-en-3-one; (17α)-17-Hydroxy-3-oxo-19-norpregn-4-ene-21-nitrile; Dienogest EP Impurity F; 2-((8R,9S,10R,13S,14S,17R)-17-Hydroxy-13-methyl-3-oxo-2,3,6,7,8,9,10,11,12,13,14,15,16,17-tetradecahydro-1H-cyclopenta[a]phenanthren-17-yl)acetonitrile. Grades: ≥95%. CAS No. 67473-36-3. Molecular formula: C20H27NO2. Mole weight: 313.43. | |
17-Desethynyl 17-Dibromomethylaceto-norethindrone Acetate Quick inquiry Where to buy Suppliers range | 17-Desethynyl 17-Dibromomethylaceto-norethindrone Acetate is an intermediate of Norethindrone, which is an oral contraceptive involved in the inhibition of cytosolic sulfotransferases. Synonyms: 17-Dibromomethylaceto-19-norpregn-4-ene-3,20-dione; Norethindrone Acetate Impurity 13; (17α)-21,21-Dibromo-3,20-dioxo-19-norpregn-4-en-17-yl acetate; (8R,9S,10R,13S,14S,17S)-17-(2,2-dibromoacetyl)-13-methyl-3-oxo-2,3,6,7,8,9,10,11,12,13,14,15,16,17-tetradecahydro-1H-cyclopenta[a]phenanthren-17-yl acetate; Estr-4-en-3-one, 17-(acetyloxy)-17-(2,2-dibromoacetyl)-, (17β)-. Grades: ≥95%. CAS No. 40228-41-9. Molecular formula: C22H28Br2O4. Mole weight: 516.26. | |
17-epi-Norethindrone (Impurity G) Quick inquiry Where to buy Suppliers range | An impurity of Norethindrone, which is an oral contraceptive involved in the inhibition of cytosolic sulfotransferases. Uses: Contraceptives, oral, synthetic. Synonyms: 17-epi-Norethindrone; 17-Hydroxy-19-norpregn-4-en-20-yn-3-one; 18-Methyllevonorgestrel; Norethisterone Impurity G (EP); Norethindrone EP Impurity G. Grades: > 95%. CAS No. 38673-36-8. Molecular formula: C20H26O2. Mole weight: 298.43. | |
17-O-Trimethylsilyl 6,7-Dehydro Norethindrone Quick inquiry Where to buy Suppliers range | 17-O-Trimethylsilyl 6,7-Dehydro Norethindrone is an impurity of Norethindrone, which is an oral contraceptive involved in the inhibition of cytosolic sulfotransferases. Uses: Tibolone intermediate. Synonyms: (17α)-17-[(Trimethylsilyl)oxy]-19-norpregna-4,6-dien-20-yn-3-one; 19-Norpregna-4,6-dien-20-yn-3-one, 17-[(trimethylsilyl)oxy]-, (17α)-; Tibolone Impurity 12. Grades: 98%. CAS No. 300542-58-9. Molecular formula: C23H32O2Si. Mole weight: 368.58. | |
17-O-Trimethylsilyl Norethindrone Quick inquiry Where to buy Suppliers range | 17-O-Trimethylsilyl Norethindrone is a derivative of Norethindrone, which is an oral contraceptive involved in the inhibition of cytosolic sulfotransferases. Synonyms: (17α)-17-[(Trimethylsilyl)oxy]-19-norpregn-4-en-20-yn-3-one; 17-(Trimethylsiloxy)-19-nor-17α-pregn-4-en-20-yn-3-one. Grades: 98%. CAS No. 28426-43-9. Molecular formula: C23H34O2Si. Mole weight: 370.60. | |
(1S)-3-Hydroxy Bortezomib Quick inquiry Where to buy Suppliers range | (1S)-3-Hydroxy Bortezomib is a metabolite of Bortezomib (B675700), the first proteasome inhibitor to be approved by the US FDA for multiple myeloma, a blood cancer. Bortezomib is a reversible inhibitor of the 26S proteasome-a barrel-shaped multiprotein particle found in the nucleus and cytosol of all eukaryotic cells. Group: Biochemicals. Grades: Highly Purified. Pack Sizes: 500ug, 5mg. Molecular Formula: C19H25BN4O5, Molecular Weight: 400.24. US Biological Life Sciences. | Worldwide |
(1S)-3-Hydroxy Bortezomib-d8 Quick inquiry Where to buy Suppliers range | (1S)-3-Hydroxy Bortezomib-d8 is labelled (1S)-3-Hydroxy Bortezomib (H818155) which is a metabolite of Bortezomib (B675700), the first proteasome inhibitor to be approved by the US FDA for multiple myeloma, a blood cancer. Bortezomib is a reversible inhibitor of the 26S proteasome-a barrel-shaped multiprotein particle found in the nucleus and cytosol of all eukaryotic cells. Group: Biochemicals. Grades: Highly Purified. Pack Sizes: 1mg, 10mg. Molecular Formula: C19H17D8BN4O5, Molecular Weight: 408.29. US Biological Life Sciences. | Worldwide |
2-[(2-Pyrazinylcarbonyl)-Bortezomib Quick inquiry Where to buy Suppliers range | 2-[(2-Pyrazinylcarbonyl)-Bortezomib is a derivative of Bortezomib (B675700) which is the first proteasome inhibitor to be approved by the US FDA for multiple myeloma, a blood cancer. Bortezomib is a reversible inhibitor of the 26S proteasome-a barrel-shaped multiprotein particle found in the nucleus and cytosol of all eukaryotic cells. Group: Biochemicals. Grades: Highly Purified. Pack Sizes: 1mg, 5mg. Molecular Formula: C24H27BN6O5, Molecular Weight: 490.32. US Biological Life Sciences. | Worldwide |
2-Deoxyguanosine N1-(Ethyl Acrylate) Quick inquiry Where to buy Suppliers range | 2-Deoxyguanosine N1-(Ethyl Acrylate) is an intermediate in the synthesis of 3-(2-Deoxy- β-D-erythro-pentofuranosyl)-3,5-dihydropyrimido[1,2-a]purine-6,10-dione (D235185). 3-(2-Deoxy- β-D-erythro-pentofuranosyl)-3,5-dihydropyrimido[1,2-a]purine-6,10-dione is likely an endogenous biomarker in humans and is readily generated from M1dG in liver cytosol, which involves xanthine oxidase and aldehyde oxidase. Group: Biochemicals. Grades: Highly Purified. CAS No. 895571-80-9. Pack Sizes: 5mg, 10mg. Molecular Formula: C15H19N5O6, Molecular Weight: 365.34. US Biological Life Sciences. | Worldwide |
2'-Deoxyguanosine N1-(Ethyl Acrylate) Quick inquiry Where to buy Suppliers range | 2'-Deoxyguanosine N1-(Ethyl Acrylate) is an intermediate in the synthesis of 3-(2-Deoxy-β-D-erythro-pentofuranosyl)-3,5-dihydropyrimido[1,2-a]purine-6,10-dione. 3-(2-Deoxy-β-D-erythro-pentofuranosyl)-3,5-dihydropyrimido[1,2-a]purine-6,10-dione is likely an endogenous biomarker in humans and is readily generated from M1dG in liver cytosol, which involves xanthine oxidase and aldehyde oxidase. Synonyms: 3-[2-Amino-9-(2-deoxy-β-D-erythro-pentofuranosyl)-6,9-dihydro-6-oxo-1H-purin-1-yl]-2-propenoic Acid Ethyl Ester. CAS No. 895571-80-9. Molecular formula: C15H19N5O6. Mole weight: 365.34. | |
3-(2-Deoxy- β-D-erythro-pentofuranosyl)-3,5-dihydropyrimido[1,2-a]purine-6,10-dione Quick inquiry Where to buy Suppliers range | 3-(2-Deoxy- β-D-erythro-pentofuranosyl)-3,5-dihydropyrimido[1,2-a]purine-6,10-dione is likely an endogenous biomarker in humans and is readily generated from M1dG in liver cytosol, which involves xanthine oxidase and aldehyde oxidase. Group: Biochemicals. Grades: Highly Purified. CAS No. 895571-79-6. Pack Sizes: 1mg, 5mg. Molecular Formula: C13H13N5O5. US Biological Life Sciences. | Worldwide |
3α,5α-Tetrahydronorethisterone Quick inquiry Where to buy Suppliers range | 3α,5α-Tetrahydronorethisterone is a metabolite of Norethindrone, which is an oral contraceptive involved in the inhibition of cytosolic sulfotransferases. Synonyms: Norethindrone Impurity 5; (3α,5α,17α)-19-Norpregn-20-yne-3,17-diol; 19-Nor-5α,17α-pregn-20-yne-3α,17-diol; 17α-Ethynyl-5α-estrane-3α,17β-diol; 17α-Ethynyl-5α-oestrane-3α,17β-diol. Grades: ≥95%. CAS No. 16392-60-2. Molecular formula: C20H30O2. Mole weight: 302.45. | |
4-Diethylaminobenzaldehyde Quick inquiry Where to buy Suppliers range | DEAB is a potent inhibitor of cytosolic (class 1) aldehyde dehydrogenase (ALDH) enzymes (IC50 values 0.057 μM, 1.2 μM, 3.0 μM, 1.2 μM, 0.16 μM, and 13 μM for inhibition of ALDH1A1, ALDH1A2, ALDH1A3, ALDH1B1, ALDH2, and ALDH5A1, respectively). DEAB is also an excellent substrate for ALDH3A1, and an irreversible inhibitor of ALDH7A1 (KI value 100 μM). Uses: 4-(diethylamino)benzaldehyde is a mechanism-based inhibitor for human aldehyde dehydrogenase isoenzymes. potent and reversible inhibitor of mouse and human class i aldehyde dehydrogenase. Synonyms: 4-(diethylamino)benzaldehyde. Grades: 99 %. CAS No. 120-21-8. Molecular formula: C11H15NO. Mole weight: 177.24. | |
5 β-Dihydrocortisol 21-Acetate Quick inquiry Where to buy Suppliers range | Cortisol derivatiove. Shows binding affinities for the cytosol glucocorticoid receptor. Group: Biochemicals. Alternative Names: (5 β,11 β)-21-(Acetyloxy)-11,17-dihydroxy-pregnane-3,20-dione; 11 β,17,21-Trihydroxy-5 β-pregnane-3,20-dione 21-Acetate; RU 18760. Grades: Highly Purified. CAS No. 64313-94-6. Pack Sizes: 10mg. US Biological Life Sciences. | Worldwide |
5(S),6(R)-DiHETE Quick inquiry Where to buy Suppliers range | 5(S),6(R)-DiHETE is a dihydroxy polyunsaturated fatty acid and a nonenzymatic hydrolysis product of leukotriene A4 (LTA4). Mouse liver cytosolic epoxide hydrolase catalyzes the conversion of LTA4 to 5(S),6(R)-DiHETE. 5(S),6(R)-DiHETE is a weak LTD4 receptor agonist in guinea pig lung membranes. It induces guinea pig ileum contraction with an ED50 value of 1.3 μM. Synonyms: (5S,6R,7E,9E,11Z,14Z)-5,6-dihydroxyicosa-7,9,11,14-tetraenoic acid. Grades: ≥95%. CAS No. 82948-88-7. Molecular formula: C20H32O4. Mole weight: 336.5. | |
6,10-di-Hydroxy Norethindrone Acetate Quick inquiry Where to buy Suppliers range | 6,10-di-Hydroxy Norethindrone Acetate is an impurity of Norethindrone Acetate, which is an oral contraceptive involved in the inhibition of cytosolic sulfotransferases. Synonyms: 6,10-Dihydroxy Norethindrone Acetate. Grades: 98%. Molecular formula: C22H28O5. Mole weight: 372.45. | |
6,7-Dehydro Norethindrone Acetate Quick inquiry Where to buy Suppliers range | An impurity of Norethindrone, which is an oral contraceptive involved in the inhibition of cytosolic sulfotransferases. Synonyms: 6,7-Dehydro Norethindrone Acetate; 17-Hydroxy-19-Nor-17α-pregna-4,6-dien-20-yn-3-one Acetate; ?-6(7)-Norenthindrone Acetate; Grades: > 95%. CAS No. 106765-04-2. Molecular formula: C22H26O3. Mole weight: 338.45. | |
6,7-Didehydro Norethindrone Quick inquiry Where to buy Suppliers range | An impurity of Norethindrone, which is an oral contraceptive involved in the inhibition of cytosolic sulfotransferases. Synonyms: (17α)-17-Hydroxy-19-norpregna-4,6-dien-20-yn-3-one; 17-Hydroxy-19-nor-17α-pregna-4,6-dien-20-yn-3-one; 7α-Ethynyl-17β-hydroxyestra-4,6-dien-3-one; 6,7-Dehydronorethindrone; Norethindrone EP Impurity A. Grades: > 95%. CAS No. 31528-46-8. Molecular formula: C20H24O2. Mole weight: 296.41. | |
6-alpha-Hydroxy Norethindrone Acetate Quick inquiry Where to buy Suppliers range | An impurity of Norethindrone, which is an oral contraceptive involved in the inhibition of cytosolic sulfotransferases. Synonyms: 6α-Hydroxy Norethindrone Acetate; (6α,17α)-17-(Acetyloxy)-6-hydroxy-19-norpregn-4-en-20-yn-3-one. Grades: > 95%. CAS No. 6856-28-6. Molecular formula: C22H28O4. Mole weight: 356.47. | |
6β,17-Norethindrone Diacetate Quick inquiry Where to buy Suppliers range | 6β,17-Norethindrone Diacetate is an impurity of Norethindrone Acetate, which is an oral contraceptive involved in the inhibition of cytosolic sulfotransferases. Synonyms: (6β,17α)-17-(Acetyloxy)-6-acetyl-19-norpregn-4-en-20-yn-3-one. Grades: 95%. Molecular formula: C24H30O4. Mole weight: 382.49. | |
6-Beta-Hydroxy-19-Norandrostenedione Quick inquiry Where to buy Suppliers range | An impurity of Norethindrone, which is an oral contraceptive involved in the inhibition of cytosolic sulfotransferases. Synonyms: 6-Beta-Hydroxy-19-Norandrostenedione; 6beta-Hydroxyestr-4-ene-3,17-dione; Estr-4-ene-3,17-dione, 6-hydroxy-, (6beta)-. Grades: > 95%. CAS No. 5949-49-5. Molecular formula: C18H24O3. Mole weight: 288.39. | |
6-beta-Hydroxy Norethindrone Acetate (Norethindrone Acetate Impurity F) Quick inquiry Where to buy Suppliers range | An impurity of Norethindrone, which is an oral contraceptive involved in the inhibition of cytosolic sulfotransferases. Synonyms: (6β,17α)-17-(Acetyloxy)-6-hydroxy-19-norpregn-4-en-20-yn-3-one; 6β,17-Dihydroxy-19-nor-17α-pregn-4-en-20-yn-3-one 17-Acetate. Grades: > 95%. CAS No. 6856-27-5. Molecular formula: C22H28O4. Mole weight: 356.47. | |
6-beta-Hydroxy Norethindrone (Norethindrone Impurity H) Quick inquiry Where to buy Suppliers range | An impurity of Norethindrone, which is an oral contraceptive involved in the inhibition of cytosolic sulfotransferases. Synonyms: 6β-Hydroxy Norethindrone; (6β,17α)-6,17-Dihydroxy-19-norpregn-4-en-20-yn-3-one; 6β,17β-Dihydroxy-17α-ethynylestr-4-en-3-one; 6β,17β-Dihydroxy-19-nor-17α-pregn-4-en-20-yn-3-one; 6β-Hydroxynorethindrone; 6β-Hydroxynorethisterone. Grades: > 95%. CAS No. 51724-44-8. Molecular formula: C20H26O3. Mole weight: 314.45. | |
6-Ketocholestanol (5a-Cholestan-6-one) Quick inquiry Where to buy Suppliers range | An oxygenated cholesterol which can be used as a ligand for cytosolic-nuclear tumor promoter binding protein. Group: Biochemicals. Alternative Names: 5a-Cholestan-6-one. Grades: Highly Purified. Pack Sizes: 1g. US Biological Life Sciences. | Worldwide |
6-Keto Norethindrone Acetate (Norethindrone Impurity G) Quick inquiry Where to buy Suppliers range | An impurity of Norethindrone, which is an oral contraceptive involved in the inhibition of cytosolic sulfotransferases. Synonyms: 6-Oxo Norethindrone Acetate; (17α)-17-(Acetyloxy)-19-norpregn-4-en-20-yne-3,6-dione; 6-Ketonorethindrone Acetate; Norethindrone Acetate EP Impurity G. Grades: > 95%. CAS No. 438244-27-0. Molecular formula: C22H26O4. Mole weight: 354.45. | |
6-Oxo Norethindrone Quick inquiry Where to buy Suppliers range | 6-Oxo Norethindrone is an impurity of Norethindrone, which is an oral contraceptive involved in the inhibition of cytosolic sulfotransferases. Synonyms: (17α)-17-Hydroxy-19-norpregn-4-en-20-yne-3,6-dione; 17α-Hydroxy-19-norpregn-4-en-20-yne-3,6-dione; 6-Ketonorethindrone. Grades: 95%. CAS No. 67696-78-0. Molecular formula: C20H24O3. Mole weight: 312.40. | |
7,8,9,10-Tetrahydro-benzo[a]pyren-7-ol Quick inquiry Where to buy Suppliers range | 7,8,9,10-Tetrahydro-benzo[a]pyren-7-ol is a Benzopyrene (B205800) derivative, activated by hepatic cytosol. Group: Biochemicals. Alternative Names: (RS) -7, 8, 9, 10-Tetrahydrobenzo [a]pyren-7-ol; (±) -7, 8, 9, 10-Tetrahydrobenzo [a]pyren-7-ol; 7-Hydroxy-7, 8, 9, 10-tetrahydrobenzo [a]pyrene; NSC 30871. Grades: Highly Purified. CAS No. 6272-55-5. Pack Sizes: 100mg. US Biological Life Sciences. | Worldwide |
9,10-Dehydro-19-nortestosterone Quick inquiry Where to buy Suppliers range | Gestagenic Testosterone derivative. A steroid ligand for the cytosol androgen receptor (AR) of rat prostate. Group: Biochemicals. Alternative Names: 17 β-Hydroxyestra-4,9-dien-3-one; 3-Oxo-4,9-estradien-17 β-ol; 17 β-hydroxy-estra-4,9-dien-3-one; 4,9-Estradien-17 β-ol-3-one; RU 3118. Grades: Highly Purified. CAS No. 6218-29-7. Pack Sizes: 100mg. US Biological Life Sciences. | Worldwide |
AACOCF Quick inquiry Where to buy Suppliers range | AACOCF, an anlogue of arachidonic acid, is a slow-binding inhibitor of cytosolic (85 kDa) phospholipase A2. It also inhibits fatty acid amide hydrolase (FAAH, anandamide amidase) in vitro. Synonyms: 1,1,1-Trifluoro-6Z,9Z,12Z,15Z-heneicosateraen-2-one; Arachidonyl trifluoromethyl ketone; Arachidonyltrifluoromethane. CAS No. 149301-79-1. Molecular formula: C21H31F3O. Mole weight: 356.47. | |
ABT 702 Quick inquiry Where to buy Suppliers range | ABT 702 is a non-nucleoside adenosine kinase (ADK) inhibitor (IC50 = 2 nM and 50 nM in cytosolic and intact cell assays, respectively). Study conformed that ABT702 could reduce pain and inflammation in animal models, yet be clastogenic in an in vitro Chinese Hamster micronucleus assay. Synonyms: ABT 702; ABT702; ABT-702; 5-(3-bromophenyl)-7-(6-morpholin-4-ylpyridin-3-yl)pyrido[2,3-d]pyrimidin-4-amine. Grades: 99%. CAS No. 214697-26-4. Molecular formula: C22H19BrN6O. Mole weight: 463.33. | |
Adenosine 3,5-cyclic Monophosphorothioate, Sp-Isomer, Triethylammonium Salt (Adenosine 3,5-cyclic Phosphorothioate-Sp, Sp-cAMPS, TEA) Quick inquiry Where to buy Suppliers range | A cell-permeable cAMP analog that binds cAMP-receptor proteins. Induces the guanine-nucleotide exchange factor activity of GEFI (also known as Epac) and GEFII towards Raf1, both in vivo and in vitro. Known to cause a decrease in cytosolic pH.CAS No.71774-13-5. Group: Biochemicals. Grades: Highly Purified. CAS No. 71774-13-5. Pack Sizes: 10umol. Molecular Formula: C??H??N?O?PS · (CH?CH?)?NH. US Biological Life Sciences. | Worldwide |
AG 205 Quick inquiry Where to buy Suppliers range | AG 205 is a progesterone receptor membrane component 1 (Pgrmc1) ligand. It inhibits cell cycle progression and cell viability in cancer cell lines. It inhibits progesterone induced cytosolic Ca2+ increases in GnRH neurons in vitro. Synonyms: Cis-2-[[1-(4-Chlorophenyl)-1H-tetrazol-5-yl]thio]-1-(1,2,3,4,4a,9b-hexahydro-2,8-dimethyl-5H-pyrido[4,3-b]indol-5-yl)-ethanone. Grades: ≥98%. CAS No. 442656-02-2. Molecular formula: C22H23ClN6OS. Mole weight: 454.98. | |
AhR Antagonist III, GNF351 (N-(2-(3H-Indol-3-yl)ethyl)-9-isopropyl-2-(5-methyl-3-pyridyl)-7H-purin-6-amine, N-(2-(1H-Indol-3-yl)ethyl)-9-isopropyl-2-(5-methylpyridin-3-yl)-9H-purin-6-amine) Quick inquiry Where to buy Suppliers range | A cell-permeable purine compound that acts as a high-affinity aryl hydrocarbon receptor (AhR) antagonist (IC50 = 62nM in mouse liver cytosol expressing humanized AhR) and lacks any agonist activity even at higher doses. Reportedly binds with high affinity to the ligand-binding pocket of AhR and blocks the binding of an array of exogenous and endogenous ligands. Shown to non-covalently interact with Ser317, His291, and Ser365 in human and with Ser311, His285, and Ser359 in mouse AhR. Represses AhR transcriptional activity via the dioxin response element (DRE)-dependent and independent mediated responses in human and mouse cells (IC50 = 8.5nM in HepG2 40/6 cells). Group: Biochemicals. Grades: Highly Purified. Pack Sizes: 10mg. US Biological Life Sciences. | Worldwide |
Antennapedia Peptide (43-58), acid Quick inquiry Where to buy Suppliers range | Antennapedia Peptide (43-58), acid, a cell-penetrating peptide corresponding to the region within the DNA binding domain of the Drosophila Antennapedia, is mapped to be responsible for cellular internalization. It is also known as penetratin and has been shown to be able to translocate through the plasma membrane to the cytosol and nucleus of living cells, both at 37°C and 4°C. Synonyms: H-Arg-Gln-Ile-Lys-Ile-Trp-Phe-Gln-Asn-Arg-Arg-Met-Lys-Trp-Lys-Lys-OH; L-arginyl-L-glutaminyl-L-isoleucyl-L-lysyl-L-isoleucyl-L-tryptophyl-L-phenylalanyl-L-glutaminyl-L-asparaginyl-L-arginyl-L-arginyl-L-methionyl-L-lysyl-L-tryptophyl-L-lysyl-L-lysine. Grades: >95%. Molecular formula: C104H168N34O20S. Mole weight: 2246.76. | |
Antennapedia Peptide(43-58) , acid Quick inquiry Where to buy Suppliers range | A peptide corresponding to the region within the Drosophila Antennapedia DNA binding domain that is mapped to be responsible for cellular internalization. This peptide is also called penetratin. The peptide has been shown to be able to translocate through the plasma membrane to the cytosol and nucleus of living cells, both at 37 ?C and 4 ?C. Uses: Antennapedia Peptides. Product ID: GR1302. | |
Antennapedia Peptide (43-58), amide Quick inquiry Where to buy Suppliers range | Antennapedia Peptide (43-58), amide, a cell-penetrating peptide corresponding to the region within the DNA binding domain of the Drosophila Antennapedia, is mapped to be responsible for cellular internalization. It is also known as penetratin and has been shown to be able to translocate through the plasma membrane to the cytosol and nucleus of living cells, both at 37°C and 4°C. Synonyms: H-Arg-Gln-Ile-Lys-Ile-Trp-Phe-Gln-Asn-Arg-Arg-Met-Lys-Trp-Lys-Lys-NH2. Grades: >95%. Molecular formula: C104H169N35O19S. Mole weight: 2245.78. | |
Antennapedia Peptide(43-58) , amide Quick inquiry Where to buy Suppliers range | A peptide corresponding to the region within the Drosophila Antennapedia DNA binding domain that is mapped to be responsible for cellular internalization. This peptide is also called penetratin. The peptide has been shown to be able to translocate through the plasma membrane to the cytosol and nucleus of living cells, both at 37 ?C and 4 ?C. Uses: Antennapedia Peptides. Product ID: GR1303. | |
Antennapedia Peptide (43-58), FAM-labeled Quick inquiry Where to buy Suppliers range | Antennapedia Peptide (43-58), FAM-labeled is an antennapedia peptide (Penetratin) labeled with FAM. It is a 16 amino acid peptide corresponding to the region within the Drosophila Antennapedia DNA binding domain that is mapped to be responsible for cellular internalization. It has been shown to be able to translocate through the plasma membrane to the cytosol and nucleus of living cells, both at 37°C and 4°C. Synonyms: 5-FAM-Arg-Gln-Ile-Lys-Ile-Trp-Phe-Gln-Asn-Arg-Arg-Met-Lys-Trp-Lys-Lys-NH2. Grades: >95%. Molecular formula: C125H179N35O25S. Mole weight: 2604.08. | |
Antennapedia Peptide(43-58) , FAM-labeled Quick inquiry Where to buy Suppliers range | This is a Antennapedia peptide(Penetratin) labeled with FAM is mapped to be responsible for cellular internalization. This peptide has been shown to be able to translocate through the plasma membrane to the cytosol and nucleus of living cells, both at 37 ?C and 4 ?C. Uses: Antennapedia Peptides. Product ID: GR1304. | |
ASB14780 Quick inquiry Where to buy Suppliers range | ASB14780 is a potent and oral inhibitor of cytosolic phospholipase A2α (cPLA2α; IC50 = 0.020 μM in vitro and 0.54 - 0.64 μM in whole blood assay) with anti-inflammatory property in ear edema and asthma models. ASB14780 has the potential for the treatment of nonalcoholic fatty liver diseases including fatty liver and hepatic fibrosis. ASB14780 significantly attenuated expression of smooth muscle a-actin (a-SMA) protein and the mRNA expression of collagen 1a2, a-SMA and TGFb1 in the liver, as well as the expression of monocyte/macrophage markers. Synonyms: ASB14780; ASB 14780; ASB-14780; 3-(3-Phenethyl-1-(4-phenoxyphenyl)-1H-indol-5-yl)propanoic acid, 2-amino-2-(hydroxymethyl)-1,3-propanediol; 3-[1-(4-Phenoxyphenyl)-3-(2-phenylethyl)-1H-indol-5-yl]propanoic acid, 2-amino-2-(hydroxymethyl)-1,3-propanediol. Grades: 99%. CAS No. 1069046-00-9. Molecular formula: C31H27NO3.C4H11NO3. Mole weight: 582.69. | |
Auranofin Quick inquiry Where to buy Suppliers range | Auranofin appears to induce heme oxygenase 1 (HO-1) mRNA, as an inhibitor of thioredoxin reductase (TrxR) (IC50 = 20 nM; Ki = 4 nM for the NADPH-reduced form of human cytosolic TrxR). Uses: Auranofin inhibits various leukocyte activation pathways at multiple sites. Synonyms: SKF-39162; SKF-D-39162; SKF 39162; SKF D 39162; SKFD-39162; SKFD39162; Ridaura; NSC 321521, Ridauragold thiol; Gold, [1-(thio-κS)-β-D-glucopyranose 2,3,4,6-tetraacetato](triethylphosphine)-; [1-(Thio-κS)-β-D-glucopyranose 2, 3, 4, 6-tetraacetato] (triethylphosphine)gold; Gold, (1-thio-β-D-glucopyranosato)(triethylphosphine)-, 2,3,4,6-tetraacetate; Gold, (1-thio-β-D-glucopyranose 2,3,4,6-tetraacetato-S)(triethylphosphine)-; β-D-Glucopyranose, 1-thio-, 2,3,4,6-tetraacetate, gold complex; [ (Tetra-O-acetyl-β -D-glucopyranosyl)thio] (triethylphosphine)gold; Aktil; Crisinor; Crisofin Gold Salt; Ridauran; SKF 39162D. Grades: ≥98%. CAS No. 34031-32-8. Molecular formula: C20H34AuO9PS. Mole weight: 678.49. | |
AX 048 Quick inquiry Where to buy Suppliers range | Ethyl 4-[(2-oxohexadecanoyl)amino]butanoate (AX 048) is a PLA2 (Phospholipase A2) and PGE2 (Prostaglandin E2) inhibitor. PLA2 is known as calcium-dependent cytosolic PLA2 (cPLA2), which selectively releases arachidonic acid from membrane phospholipids. It plays a central role in initiating the synthesis of prostaglandins and leukotrienes. This compound also contains a specific affinity for group IVA cPLA2 which moderates antihyperalgesia effects. Synonyms: AX-048; AX 048; Butanoic acid, 4-((1,2-dioxohexadecyl)amino)-, ethyl ester; UNII-8782Z45DLV; 8782Z45DLV; Butanoic acid, 4-[(1,2-dioxohexadecyl)amino]-, ethyl ester; ethyl 4-(2-oxohexadecanoylamino)butanoate; ethyl 4-(2-oxohexadecanamido)butanoate; CHEMBL574723; SCHEMBL4781039; DTXSID60236282; AKOS040755666; ethyl 4-[(2-oxohexadecanoyl)amino] butanoate; Q27269809; 4- [(1, 2- dioxohexadecyl)amino]- butanoic acid, ethyl ester. Grades: ≥98%. CAS No. 873079-69-7. Molecular formula: C22H41NO4. Mole weight: 383.6. | |
b-AP15 Quick inquiry Where to buy Suppliers range | b-AP15 is a deubiquitinases inhibitor for 19S proteasomes activity of Ub-AMC cleavage with IC50 of 2.1 μM.Not a general deubiquitinase inhibitor. Has minimal inhibition on recombinant and cytosolic nonproteasomal cysteine deubiquitinases. Synonyms: b-AP15; b-AP15; b-AP-15; USP14 Inhibitor III; UCHL5UCH37 Inhibitor II; NSC687852. Grades: >98%. CAS No. 1009817-63-3. Molecular formula: C22H17N3O6. Mole weight: 419.39. | |
BCATc Inhibitor 2 Quick inquiry Where to buy Suppliers range | BCATc Inhibitor 2 is a sulfonyl hydrazide that inhibits BCATc with IC50s of 0.81 for human and IC50 s of 0.2 μM for rat. It is 15-fold selectivity over BCATm. It has also been used to block calcium influx into neurons with IC50 of 4.8 μM following inhibition of glutamate uptake and to demonstrate neuroprotective efficacy in an in vivo rat model of neurodegeneration. Synonyms: Cytosolic Branched-Chain Amino Acid Transferase Inhibitor 2. Grades: ≥98%. CAS No. 406191-34-2. Molecular formula: C16H10ClF3N2O4S. Mole weight: 418.8. | |
BGT226 Quick inquiry Where to buy Suppliers range | BGT226 is a phosphatidylinositol 3-kinase (PI3K) inhibitor with potential antineoplastic activity. BGT226 specifically inhibits PIK3 in the PI3K/AKT kinase (or protein kinase B) signaling pathway, which may trigger the translocation of cytosolic Bax to the mitochondrial outer membrane, increasing mitochondrial membrane permeability. Synonyms: BGT-226; BGT 226; BGT-226 free base; BGT226 free base; NVP-BGT226; 1,3-Dihydro-8-(6-methoxy-3-pyridinyl)-3-methyl-1-[4-(1-piperazinyl)-3-(trifluoromethyl)phenyl]-2H-imidazo[4,5-c]quinolin-2-one. Grades: 98%. CAS No. 915020-55-2. Molecular formula: C32H29F3N6O6. Mole weight: 534.54. | |
BMS-229724 Quick inquiry Where to buy Suppliers range | BMS-229724 is a selective tight-binding inhibitor of cytosolic phospholipase A2 (cPLA2) in that it did not inhibit secreted phospholipase A2 in vitro, nor phospholipase C and phospholipase D in cells. BMS-22972 acts at the lipid/water interface and possesses anti-inflammatory activity in skin inflammation models. Synonyms: 4-[4-[2-[2-[bis (4-chlorophenyl) methoxy]ethylsulfonyl]ethoxy]phenyl]-1, 1, 1-trifluorobutan-2-one; 4- (4- (2- (2- (bis (4-chlorophenyl) methoxy) ethylsulfonyl) ethoxy) phenyl) -1, 1, 1-trifluoro-2-butanone; BMS-229724; BMS 229724; BMS229724; 42AD6D8ECA; SCHEMBL3304414; LS-46643; UNII-42AD6D8ECA. Grades: >98%. CAS No. 221914-85-8. Molecular formula: C27H25Cl2F3O5S. Mole weight: 589.45. | |
Bortezomib, deuterated (Velcade-deuterated, [ (1R) -3-Methyl-1- [ [ (2S) -1-oxo-3-phenyl-2- [ (pyrazinylcarbonyl) amino] propyl] amino] butyl] -boronic Acid-deuterated) Quick inquiry Where to buy Suppliers range | Bortezomib is the first proteasome inhibitor to be approved b the US FDA for multiple myeloma, a blood cancer. A reversible inhibitor of the 26S proteasome-a barrel-shaped multiprotein particle found in the nucleus and cytosol of all eukaryotic cells. Group: Biochemicals. Alternative Names: Velcade-deuterated, [ (1R) -3-Methyl-1- [ [ (2S) -1-oxo-3-phenyl-2- [ (pyrazinylcarbonyl) amino] propyl] amino] butyl] -boronic Acid-deuterated. Grades: Highly Purified. Pack Sizes: 1mg. US Biological Life Sciences. | Worldwide |
Bromoenol lactone Quick inquiry Where to buy Suppliers range | BEL is a selective, potent, irreversible, mechanism-based inhibitor of myocardial cytosolic calcium-independent phospholipase A2 (iPLA2) with a Ki value of 180 nM. BEL induces the proteolysis of procaspase-9 and procaspase-3 and increases cleavage of poly (ADP-ribose) polymerase. BEL also inhibits macrophage iPLA2 in a concentration-dependent manner with an IC50 value of 60 nM and is an effective enzyme-activated irreversible inhibitor of chymotrypsin Ki of 636 nM. Long term treatment with BEL increased annexin-V binding to the cell surface and nuclear DNA damage. Synonyms: BEL; Haloenol lactone; HELSS. Grades: ≥95%. CAS No. 88070-98-8. Molecular formula: C16H13BrO2. Mole weight: 317.2. | |
C16 Ceramide-1-phosphate (d18:1/16:0) ammonium salt Quick inquiry Where to buy Suppliers range | C16 Ceramide-1-phosphate (C16 C1P) is one of the main forms of C1P found in cells. It is created by phosphorylation of by ceramide kinase. It activates cytosolic phospholipase A2α (PLA2α) and stimulates the release of arachidonic acid in A549 cells. Synonyms: C16 C1P; C16 Ceramide-1-phosphate; N-(hexadecanoyl)-sphing-4-enine-1-phosphate; CerP(d18:1/16:0). Grades: ≥98%. CAS No. 1246303-22-9. Molecular formula: C34H71N2O6P. Mole weight: 634.91. | |
C16 Ceramide (N-Palmitoyl-D-Sphingosine, N-Hexadecanoyl-D-sphingosine, Palmitoyl Ceramide) Quick inquiry Where to buy Suppliers range | A predominant, rather hydrophobic natural ceramide. Activates a cytosolic serine/threonine protein phosphatase in T9 cells; induces EGF receptor phosphorylation in A-431 cells; stimulates ceramide-activated protein kinase. Group: Biochemicals. Alternative Names: N-Palmitoyl-D-Sphingosine; N-Hexadecanoyl-D-sphingosine; Palmitoyl Ceramide. Grades: Highly Purified. CAS No. 24696-26-2. Pack Sizes: 5mg. US Biological Life Sciences. | Worldwide |
cADP-Ribose (cADPR) Ammonium Salt Quick inquiry Where to buy Suppliers range | Cyclic ADP-ribose ammonium is a potent calcium-mobilized second messenger synthesized from NAD+ by ADP-ribosyl cyclase. It increases cytosolic calcium mainly by Ryanodine receptor-mediated release from endoplasmic reticulum and extracellular influx through the opening of TRPM2 channels. Synonyms: cADP-Ribose Ammonium Salt; cADPR Ammonium Salt; cyclic ADP-ribose ammonium salt; Cyclic Adenosine Diphosphate Ribose ammonium salt; Cyclic adenosine 5'-diphosphate ribose ammonium salt. Grades: 90%. Molecular formula: C15H21N5O13P2.x(NH3). Mole weight: 541.30 (free base). | |
CAY10502 Quick inquiry Where to buy Suppliers range | Phospholipases A2 (PLA2s) are enzymes that cleave fatty acid in position two of phospholipids, hydrolyzing the bond between the second fatty acid "tail" and the glycerol molecule. It catalyzes the hydrolysis of phospholipids at the sn-2 position leading to the production of lysophospholipids and free fatty acids. CAY10502 is a potent Calcium-dependent cytosolic PLA2 (cPLA2α) inhibitor with IC50 value of 4.3 nM for the purified enzyme from human platelets. It inhibits arachidonic acid mobilization from A23187-stimulated or TPA-stimulated human platelets with IC50 values of 570 and 0.9 nM, respectively. Synonyms: CAY10502; CAY-10502. Grades: ≥98% (mixture of isomers). CAS No. 888320-29-4. Molecular formula: C30H37NO7. Mole weight: 523.6. | |
CAY10590 Quick inquiry Where to buy Suppliers range | Phospholipase A2 (PLA2) catalyzes the hydrolysis of fatty acids at the sn-2 position of glycerophospholipids, liberating arachidonic acid for subsequent eicosanoid synthesis. There are three primary types of PLA2 exist: secretory (sPLA2), calcium-dependent cytosolic (cPLA2), and calcium-independent cytosolic (iPLA2). CAY10590 is a selective and potent inhibitor of sPLA2. It exhibits 95% inhibition (XI(50) = 0.003) of sPLA2 at 0.091 mole fraction without affecting the activities of cPLA2 or iPLA2. Synonyms: CAY 10590; CAY-10590. Grades: ≥98%. CAS No. 1101136-50-8. Molecular formula: C21H33NO3. Mole weight: 347.5. | |
CAY10650 Quick inquiry Where to buy Suppliers range | Cytosolic phospholipase A2α (cPLA2α) specifically catalyzes the hydrolysis of arachidonic acid from the sn-2-ester position of membrane phospholipids, playing a central role in initiating the synthesis of prostaglandins and leukotrienes, both important mediators of the inflammatory process. CAY10650 is a highly potent (IC50 = 12 nM) cPLA2α inhibitor. It demonstrates strong anti-inflammatory effects when applied topically at a dose of 0.1 mg/ear in a mouse model of acute irritant contact dermatitis. Synonyms: CAY 10650; CAY-10650. Grades: >98%. CAS No. 1233706-88-1. Molecular formula: C28H25NO6. Mole weight: 471.5. | |
CCT 031374 hydrobromide Quick inquiry Where to buy Suppliers range | CCT 031374 hydrobromide is an inhibitor of TCF-dependent transcription. It was shown to block BIO-induced β-catenin stabilization, and reduce nuclear and cytosolic β-catenin levels in mouse L-cells. Synonyms: SR 01000418274; CCT 031374 hydrobromide; SR01000418274; CCT031374 hydrobromide; SR-01000418274; CCT-031374 hydrobromide; 1-[1,1'-Biphenyl]-4-yl-2-(2,3-dihydro-9H-imidazo[1,2-a]benzimidazol-9-yl)ethanone hydrobromide. Grades: ≥98% by HPLC. CAS No. 1219184-91-4. Molecular formula: C23H19N3O.HBr. Mole weight: 434.33. | |
CCT 031374 hydrobromide (1-[1,1'-Biphenyl]-4-yl-2-(2,3-dihydro-9H-imidazo[1,2-a]benzimidazol-9-yl)ethanone hydrobromide) Quick inquiry Where to buy Suppliers range | Inhibitor of TCF-dependent transcription. Blocks BIO-induced beta-catenin stabilization; reduces nuclear and cytosolic beta-catenin levels in mouse L-cells. Inhibits growth and reduces TCF-dependent transcription in SW480 colon carcinoma cells. Group: Biochemicals. Grades: Highly Purified. CAS No. 1219184-91-4. Pack Sizes: 10mg. US Biological Life Sciences. | Worldwide |
CDIBA Quick inquiry Where to buy Suppliers range | CDIBA is a potent and selective cytosolic phospholipase A2 (cPLA2) inhibitor. Synonyms: 4-[2-(1-benzhydryl-5-chloro-2-methylindol-3-yl)ethoxy]benzoic acid. Grades: 99%. CAS No. 479422-22-5. Molecular formula: C31H26ClNO3. Mole weight: 496. | |
Chelerythrine chloride Quick inquiry Where to buy Suppliers range | Cell permeable potent inhibitor of protein kinase C. Does not inhibit tyrosine protein kinases, cAMP-dependent protein kinase or calcium/calmodulin-dependent protein kinase. Antiplatelet, anti-inflammatory, antibacterial and antitumor compound. Apoptosis inducer in cancer cells in vitro and in vivo. Activates MAPK and JUNK signaling pathways. Affects translocation of PKC from cytosol to plasma membrane. Neurite outgrowth stimulator. Inhibits binding of BclXL to Bak (IC50 =1.5uM) or Bad proteins and stimulates apoptosis in several cancer cell lines. Blocks human P2X7 receptor. Induces cell cycle arrest in G1 phase. Specific cyclooxygenase-2 inhibitor. Group: Biochemicals. Alternative Names: NSC 36405, 1,2-Dimethoxy-N-methyl-[1,3]benzodioxolo[5,6-c]phenanthridinium chloride. Grades: Highly Purified. CAS No. 3895-92-9. Pack Sizes: 1mg, 5mg, 25mg. Molecular Formula: C21H18ClNO4. US Biological Life Sciences. | Worldwide |
Clodronate Liposome Quick inquiry Where to buy Suppliers range | Clodronate Liposome is a multilamellar liposome suspension in which clodronate is encapsulated in the aqueous compartments of the liposomes. When animals or cells are treated with Clodronate Liposome, phagocytic cells recognize the liposomes as invading foreign particles and proceed to remove the liposomes from the local tissue or serum via phagocytosis. The liposomes then release clodronate into the cytosol, resulting in cell death. Non-encapsulated clodronate cannot cross the cell membrane to initiate cell death. Group: Clodronate liposome. | |
Collismycin A Quick inquiry Where to buy Suppliers range | It is produced by the strain of Streptomyces sp. MQ22. It has the inhibitory effect of dexamethasone-glucocorticoid receptor. IC50 is 1.5 X 10-5 mol/L (rat liver cytosol). It has the anti-tumor cell activity, inhibits rat leukemia cell L1210 with IC50 of 0.08 μg/mL. Synonyms: (E)-4-Methoxy-5-(methylthio)-[2,2'-bipyridine]-6-carbaldehyde oxime; (2E)-4-methoxy-3-methylsulfanyl-2-(nitrosomethylidene)-6-pyridin-2-yl-1H-pyridine. Grades: ≥ 95%. CAS No. 158792-24-6. Molecular formula: C13H13N3O2S. Mole weight: 275.33. | |
Collismycin B Quick inquiry Where to buy Suppliers range | It is produced by the strain of Streptomyces sp. MQ22. It has the inhibitory effect of dexamethasone-glucocorticoid receptor. IC50 is 1.0 X 10-5 mol/L (rat liver cytosol). It has the anti-tumor cell activity, inhibits rat leukemia cell L1210 with IC50 of 0.12 μg/mL. Synonyms: (2Z)-4-methoxy-3-methylsulfanyl-2-(nitrosomethylidene)-6-pyridin-2-yl-1H-pyridine; 4-methoxy-3-methylsulfanyl-2-(nitrosomethylene)-6-(2-pyridyl)-1H-pyridine. CAS No. 158792-25-7. Molecular formula: C13H13N3O2S. Mole weight: 275.33. | |
Conduritol B epoxide Quick inquiry Where to buy Suppliers range | Conduritol B epoxide (CBE) is an irreversible inhibitor of covalently bound acid β-glucosidase, also known as GBA, or GBA1 (IC50 = 9 μM). It also does not inhibit non-lysosomal glucosylceramidase or cytosolic β-glucosidase. Synonyms: CBE; 1,2-anhydro-myo-inositol. Grades: ≥95%. CAS No. 6090-95-5. Molecular formula: C6H10O5. Mole weight: 162.1. |