Noradrenaline Suppliers USA

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Product
Noradrenaline bitartrate Noradrenaline bitartrate. Group: Biochemicals. Grades: Purified. CAS No. 108341-18-0. Pack Sizes: 50mg. US Biological Life Sciences. USBiological 5
Worldwide
Noradrenaline bitartrate Noradrenaline bitartrate. Uses: For analytical and research use. Group: Impurity standards. CAS No. 69815-49-2. Molecular Formula: C12H19NO10. Mole Weight: 337.28. Catalog: APB69815492. Alfa Chemistry Analytical Products 3
Noradrenaline bitartrate monohydrate Noradrenaline bitartrate monohydrate is a direct alpha-adrenergic receptors stimulator. Noradrenaline modulates the gain of evoked activity, especially in sensory areas. Synonyms: 4-[(1R)-2-Amino-1-hydroxyethyl]-1,2-benzenediol Hydrogen Tartrate Monohydrate; L-Noradrenaline Bitartrate Monohydrate; Levoarterenol Bitartrate Monohydrate; L-Arterenol Bitartrate Monohydrate; 1,2-Benzenediol, 4-[(1R)-2-amino-1-hydroxyethyl]-, (2R,3R)-2,3-dihydroxybutanedioate, hydrate (1:1:1); 1,2-Benzenediol, 4-(2-amino-1-hydroxyethyl)-, (R)-, [R-(R*,R*)]-2,3-dihydroxybutanedioate (1:1) (salt), monohydrate; Arterenol, tartrate, monohydrate. Grades: >98%. CAS No. 108341-18-0. Molecular formula: C12H19NO10. Mole weight: 337.28. BOC Sciences 9
DL-Noradrenaline hydrochloride 5g Pack Size. Group: Bioactive Small Molecules, Biochemicals, Research Organics & Inorganics. Formula: C8H11NO3 · HCl. CAS No. 55-27-6. Prepack ID 37506482-5g. Molecular Weight 205.64. See USA prepack pricing. Molekula Americas
L-Noradrenaline 100mg Pack Size. Group: Bioactive Small Molecules, Biochemicals, Research Organics & Inorganics. Formula: C8H11NO3. CAS No. 51-41-2. Prepack ID 90028019-100mg. Molecular Weight 169.18. See USA prepack pricing. Molekula Americas
L-Noradrenaline 1g Pack Size. Group: Bioactive Small Molecules, Biochemicals, Research Organics & Inorganics. Formula: C8H11NO3. CAS No. 51-41-2. Prepack ID 90028019-1g. Molecular Weight 169.18. See USA prepack pricing. Molekula Americas
L-Noradrenaline Norepinephrine is the US name for noradrenaline, a catecholamine with multiple roles including as a hormone and a neurotransmitter. It performs its action by being released into the synaptic cleft, where it acts on adrenergic receptors, followed by the signal termination, either by degradation of norepinephrine, or by uptake by surrounding cells. Uses: Adrenergic alpha-agonists. Synonyms: (R)-4-(2-Amino-1-hydroxyethyl)-1,2-benzenediol; l-Arterenol; (-)-α-(Aminomethyl)-3,4-dihydroxy-benzyl Alcohol; 4-[(1R)-2-Amino-1-hydroxyethyl]-1,2-benzenediol; (-)-Arterenol; (-)-Noradrenaline; (-)-Norepinephrine; (-)-α-(Aminomethyl)protocatechuyl Alcohol; (R)-(-)-Norepinephrine; (R)-Noradrenaline; (R)-Norepinephrine; Adrenor; Aktamin; Arterenol; Levarterenol; Levoarterenol; Levonor; Levonoradrenaline; Levonorepinephrine; Levophed; Nor-Epirenan; Noradrenalin; Noradrenaline; Norartrinal; Norepinephrine; Norepirenamine; Sympathin E; l-1-(3,4-Dihydroxyphenyl)-2-aminoethanol; l-2-Amino-1-(3,4-dihydroxyphenyl)ethanol; l-3,4-Dihydroxyphenylethanolamine; l-Arterenol; l-Noradrenaline; l-Norepinephrine; l-α-(Aminomethyl)-3,4-dihydroxybenzyl Alcohol. Grades: >98%. CAS No. 51-41-2. Molecular formula: C8H11NO3. Mole weight: 169.18. BOC Sciences 11
L-Noradrenaline hydrochloride 1g Pack Size. Group: Bioactive Small Molecules, Biochemicals, Research Organics & Inorganics. Formula: C8H11NO3 · HCl. CAS No. 329-56-6. Prepack ID 30542591-1g. Molecular Weight 205.64. See USA prepack pricing. Molekula Americas
(+)-Noradrenaline Bitartrate (+)-Noradrenaline Bitartrate is an agonist at α1- and α2-adrenoreceptors. Synonyms: (S)-4-(2-Amino-1-hydroxyethyl)-1,2-benzenediol [R-(R*,R*)]-2,3-Dihydroxybutanedioate (1:1) (salt); 4-[(1S)-2-Amino-1-hydroxyethyl]-1,2-benzenediol (2R,3R)-2,3-Dihydroxybutanedioate (1:1) (salt); α-(Aminomethyl)-3,4-dihydroxy-benzyl Alcohol (+)-Tartrate (1:1); (+)-(S)-Norepinephrine Bitartrate; (+)-Noradrenaline (+)-Bitartrate; (+)-Norepinephrine (+)-Bitartrate; (+)-Norepinephrine Bitartrate; D-Norepinephrine Bitartrate; D-Norepinephrine d-Bitartrate; S-(+)-Norepinephrine Bitartrate; d-Noradrenaline Bitartrate; d-Noradrenaline Hydrogen Tartrate; (S)-4-(2-Amino-1-hydroxyethyl)benzene-1,2-diol (2R,3R)-2,3-Dihydroxysuccinate. Grades: ≥95%. CAS No. 636-88-4. Molecular formula: C12H17NO9. Mole weight: 469.35. BOC Sciences 8
Norepinephrine Tartrate (Noradrenaline Tartrate) A derivative of Epinephrine. Epinephrine is a natural neurotransmitter that is released from the adrenal medulla and activates adrenoceptors. Synonyms: Noradrenaline Tartrate; 1,2-Benzenediol, 4-[(1R)-2-amino-1-hydroxyethyl]-, 2,3-dihydroxybutanedioate. Grades: > 95%. CAS No. 339091-66-6. Molecular formula: C8H11NO3. C4H6O6. Mole weight: 319.26. BOC Sciences 8
1,1'-(4,5-Dihydroxy-1,2-(phenylene-d2))bis-ethanone 1,1'-(4,5-Dihydroxy-1,2-(phenylene-d2))bis-ethanone is an intermediate in the synthesis of (+)-Noradrenaline-d6 Bitartrate (N661027), which is a labeled analogue of (+)-Noradrenaline Bitartrate (N661025), an agonist at α1- and α2-adrenoreceptors. Group: Biochemicals. Grades: Highly Purified. Pack Sizes: 1mg, 2.5mg. Molecular Formula: C10H8D2O4. US Biological Life Sciences. USBiological 9
Worldwide
1- (2-Cyano-1- (4-methoxyphenyl) ethyl) cyclohexanol-d6 A deuterated intermediate in the synthesis of the metabolite of Venlafaxine, a selective serotonin noradrenaline reuptake inhibitor. Used as an antidepressant. Group: Biochemicals. Grades: Highly Purified. Pack Sizes: 5mg. US Biological Life Sciences. USBiological 1
Worldwide
1-(3,4-Dihydroxyphenyl)-2-[(phenylmethyl)amino]-ethanone-d5 1-(3,4-Dihydroxyphenyl)-2-[(phenylmethyl)amino]-ethanone-d5 is an intermediate in the synthesis of (+)-Noradrenaline-d6 Bitartrate (N661027), which is a labeled analogue of (+)-Noradrenaline Bitartrate (N661025), an agonist at α1- and α2-adrenoreceptors. Group: Biochemicals. Grades: Highly Purified. Pack Sizes: 2.5mg, 5mg. Molecular Formula: C15H10D5NO3. US Biological Life Sciences. USBiological 9
Worldwide
1400W dihydrochloride (N- (3- (Aminomethyl) benzyl) acetamidine. 2HCl) A slow, tight binding and highly selective inhibitor of iNOS (inducible nitric oxide synthase/NOS II) (Kd < 7 nM). Weak and reversible inhibition of nNOS (neuronal nitric oxide synthase/NOS I) (Ki < 2) and eNOS (endothelial nitric oxide synthase/NOS III) (Ki < 50 µM). Inhibits tumor growth. Increases vasoconstriction to noradrenaline. Improves contractile function. Improves stroke outcome and decreases glutamate release. Anti-inflammatory. Group: Biochemicals. Alternative Names: N- (3- (Aminomethyl) benzyl) acetamidine. 2HCl. Grades: Highly Purified. CAS No. 214358-33-5. Pack Sizes: 5mg, 25mg, 100mg. Molecular Formula: C10H15N3. 2HCl. US Biological Life Sciences. USBiological 3
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1- (Cyano- (4-methoxyphenyl) ethyl) cyclohexanol-d10 1- (Cyano- (4-methoxyphenyl) ethyl) cyclohexanol-d10 is the labeled analogue of 1- (Cyano- (4-methoxyphenyl) ethyl) cyclohexanol (C982103), an intermediate in the synthesis of N, O-Dides methyl venlafaxine, a metabolite of Venlafaxine (V120000), a selective serotonin noradrenaline reuptake inhibitor. Used as an antidepressant. Group: Biochemicals. Grades: Highly Purified. Pack Sizes: 10mg, 100mg. Molecular Formula: C15H9D10NO2, Molecular Weight: 255.38. US Biological Life Sciences. USBiological 9
Worldwide
1-Fluoronaphthalene 1-Fluoronaphthalene is an organofluorine compound derived from naphthalene derivatives and fluorinated aromatics. 1-Fluoronaphthalene can be used to synthesize LY248686, a potent inhibitor of serotonin and noradrenaline uptake [1]. Uses: Scientific research. Group: Signaling pathways. CAS No. 321-38-0. Pack Sizes: 10 mM * 1 mL; 25 g. Product ID: HY-32126. MedChemExpress MCE
2- (1-Hydroxycyclohexyl) -2- (3- ( ( (2- (1-hydroxycyclohexyl) -2- (4-methoxyphenyl) ethyl) amino) methyl) -4-methoxyphenyl) acetonitrile 2- (1-Hydroxycyclohexyl) -2- (3- ( ( (2- (1-hydroxycyclohexyl) -2- (4-methoxyphenyl) ethyl) amino) methyl) -4-methoxyphenyl) acetonitrile is an intermediate in the synthesis of O-Desmethyl Venlafaxine N-Dimer is a dimer impurity of O-Desmethyl Venlafaxine (D296500); a metabolite of Venlafaxine (V120000) which is a selective serotonin noradrenaline reuptake inhibitor (SNRI). Also used as an antidepressant. Group: Biochemicals. Grades: Highly Purified. Pack Sizes: 10mg, 25mg. Molecular Formula: C31H42N2O4. US Biological Life Sciences. USBiological 9
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2- (3-Formyl-4-methoxyphenyl) -2- (1-hydroxycyclohexyl) acetonitrile 2- (3-Formyl-4-methoxyphenyl) -2- (1-hydroxycyclohexyl) acetonitrile is an intermediate in the synthesis of O-Desmethyl Venlafaxine N-Dimer is a dimer impurity of O-Desmethyl Venlafaxine (D296500); a metabolite of Venlafaxine (V120000) which is a selective serotonin noradrenaline reuptake inhibitor (SNRI). Also used as an antidepressant. Group: Biochemicals. Grades: Highly Purified. Pack Sizes: 10mg, 25mg. Molecular Formula: C16H19NO3. US Biological Life Sciences. USBiological 9
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2-Amino-1-phenylethanol 2-Amino-1-phenylethanol is an analogue of noradrenaline. Uses: Scientific research. Group: Natural products. CAS No. 7568-93-6. Pack Sizes: 10 mM * 1 mL; 500 mg; 1 g. Product ID: HY-59132. MedChemExpress MCE
2-[Bis (phenylmethyl)amino]-1- (3, 4-dimethoxyphenyl)-ethanone 2-[Bis (phenylmethyl)amino]-1- (3, 4-dimethoxyphenyl)-ethanone is an intermediate in synthesizing (+)-Noradrenaline-d6 Bitartrate (N661027) which is a labeled analogue of (+)-Noradrenaline Bitartrate (N661027), an agonist at α1- and α2-adrenoreceptors. Group: Biochemicals. Grades: Highly Purified. CAS No. 30332-44-6. Pack Sizes: 10mg, 25mg. Molecular Formula: C24H25NO3, Molecular Weight: 375.46. US Biological Life Sciences. USBiological 9
Worldwide
2-Bromo-4- ( (tert-butyldimethylsilyl) oxy) phenol 2-Bromo-4- ( (tert-butyldimethylsilyl) oxy) phenol is an intermediate in synthesizing rac 5’-Hydroxy Reboxetine Hydrochloride (H953470), which is an hydroxylated metabolite of Reboxetine (R142000), a selective noradrenaline reuptake inhibitor and an antidepressant. Group: Biochemicals. Grades: Highly Purified. Pack Sizes: 5mg, 10mg. Molecular Formula: C12H19BrO2Si. US Biological Life Sciences. USBiological 10
Worldwide
2- (Cyclohex-1-en-1-yl-d9) -2- (4-methoxyphenyl) acetonitrile 2- (Cyclohex-1-en-1-yl-d9) -2- (4-methoxyphenyl) acetonitrile is an impurity of Venlafaxine-d10 Hydrochloride, the labeled analogue of D,L-Venlafaxine, Hydrochloride (V120000), a selective serotonin noradrenaline reuptake inhibitor. Used as an antidepressant. Group: Biochemicals. Grades: Highly Purified. Pack Sizes: 10mg, 100mg. Molecular Formula: C15H8D9NO, Molecular Weight: 236.36. US Biological Life Sciences. USBiological 9
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2-Desamino 2-Chloro Norepinephrine 2-Desamino 2-Chloro Norepinephrine is an impurity of Noradrenaline, which is widely used as an injectable drug for the treatment of critically low blood pressure. Synonyms: 4-(2-Chloro-1-hydroxyethyl)-1,2-benzenediol; α-(Chloromethyl)-3,4-dihydroxy-benzyl alcohol; 1-(3,4-Dihydroxyphenyl)-2-chloroethanol; 1,2-Benzenediol, 4-(2-chloro-1-hydroxyethyl)-; Norepinephrine Impurity 35; Noradrenaline (Norepinephrine) Impurity 13. Grades: ≥95%. CAS No. 5530-29-0. Molecular formula: C8H9ClO3. Mole weight: 188.61. BOC Sciences 8
2-(Dibenzylamino)-3',4'-dihydroxy-acetophenone 2-(Dibenzylamino)-3',4'-dihydroxy-acetophenone is an intermediate in the synthesis of (+)-Noradrenaline-d6 Bitartrate (N661027), which is a labeled analogue of (+)-Noradrenaline Bitartrate (N661025), an agonist at α1- and α2-adrenoreceptors. Group: Biochemicals. Grades: Highly Purified. CAS No. 13062-58-3. Pack Sizes: 10mg, 25mg. Molecular Formula: C22H21NO3. US Biological Life Sciences. USBiological 9
Worldwide
2-Methoxy-4- (trifluoromethyl) phenol 2-Methoxy-4- (trifluoromethyl) phenol was used for preparation of aryl oxybenzyl morpholines as dual serotonin and noradrenaline reuptake inhibitors. Group: Biochemicals. Grades: Highly Purified. CAS No. 1027888-79-4. Pack Sizes: 100mg, 250mg. Molecular Formula: C8H7F3O2, Molecular Weight: 192.14. US Biological Life Sciences. USBiological 10
Worldwide
(2R)-2-Benzoyl-4-morpholinecarboxylic Acid 1,1-Dimethylethyl Ester (2R)-2-Benzoyl-4-morpholinecarboxylic Acid 1,1-Dimethylethyl Ester is an intermediate in synthesizing rac 5’-Hydroxy Reboxetine Hydrochloride (H953470), which is an hydroxylated metabolite of Reboxetine (R142000), a selective noradrenaline reuptake inhibitor and an antidepressant. Group: Biochemicals. Grades: Highly Purified. CAS No. 869088-60-8. Pack Sizes: 25mg, 50mg. Molecular Formula: C16H21NO4. US Biological Life Sciences. USBiological 10
Worldwide
(2R)-2-[(S)-hydroxyphenylmethyl]-4-morpholinecarboxylic Acid 1,1-Dimethylethyl Ester (2R)-2-[(S)-hydroxyphenylmethyl]-4-morpholinecarboxylic Acid 1,1-Dimethylethyl Ester is an intermediate in synthesizing rac 5’-Hydroxy Reboxetine Hydrochloride (H953470), which is an hydroxylated metabolite of Reboxetine (R142000), a selective noradrenaline reuptake inhibitor and an antidepressant. Group: Biochemicals. Grades: Highly Purified. CAS No. 1030837-58-1. Pack Sizes: 10mg, 25mg. Molecular Formula: C16H23NO4. US Biological Life Sciences. USBiological 10
Worldwide
(2R) -2-[ (S) -[ (Methylsulfonyl) oxy]phenylmethyl]-4-morpholinecarboxylic Acid 1,1-Dimethylethyl Ester (2R) -2-[ (S) -[ (Methylsulfonyl) oxy]phenylmethyl]-4-morpholinecarboxylic Acid 1,1-Dimethylethyl Ester is an intermediate in synthesizing rac 5’-Hydroxy Reboxetine Hydrochloride (H953470), which is an hydroxylated metabolite of Reboxetine (R142000), a selective noradrenaline reuptake inhibitor and an antidepressant. Group: Biochemicals. Grades: Highly Purified. CAS No. 1030837-66-1. Pack Sizes: 5mg, 10mg. Molecular Formula: C17H25NO6S, Molecular Weight: 371.45. US Biological Life Sciences. USBiological 10
Worldwide
(2S,3R)-2-Amino-3-(3-(benzoyloxy)-4-hydroxyphenyl)-3-hydroxypropanoic Acid (2S,3R)-2-Amino-3-(3-(benzoyloxy)-4-hydroxyphenyl)-3-hydroxypropanoic Acid is an impurity of Droxidopa, which is a synthetic amino acid precursor used as a prodrug to the neurotransmitter norepinephrine (noradrenaline). Molecular formula: C16H15NO6. Mole weight: 317.29. BOC Sciences 8
3, 4-Dichloro-α - [ [ [ (3-methoxyphenyl) methyl] methylamino] methyl] -benzenemethanol Used in the preparation of aryltetra hydroisoquinolines as dopamine and noradrenaline reuptake inhibitors. Group: Biochemicals. Alternative Names: (+) 3, 4-Dichloro-α - [ [ [ (3-methoxyphenyl) methyl] methylamino] methyl] -benzenemethanol. Grades: Highly Purified. CAS No. 802051-24-7. Pack Sizes: 25mg. US Biological Life Sciences. USBiological 2
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3, 4-Dichloro-α - [ [ [ (3-methoxyphenyl) methyl] methylamino] methyl] -benzenemethanol-d3 Used in the preparation of aryltetra hydroisoquinolines as dopamine and noradrenaline reuptake inhibitors. Group: Biochemicals. Alternative Names: (+) 3, 4-Dichloro-α - [ [ [ (3-methoxyphenyl) methyl] methylamino] methyl] -benzenemethanol-d3. Grades: Highly Purified. Pack Sizes: 5mg. US Biological Life Sciences. USBiological 2
Worldwide
3-Bromo-4-ethoxy-phenol 3-Bromo-4-ethoxy-phenol is an intermediate in synthesizing rac 5’-Hydroxy Reboxetine Hydrochloride (H953470), which is an hydroxylated metabolite of Reboxetine (R142000), a selective noradrenaline reuptake inhibitor and an antidepressant. Group: Biochemicals. Grades: Highly Purified. CAS No. 1216224-85-9. Pack Sizes: 5mg, 10mg. Molecular Formula: C8H9BrO2. US Biological Life Sciences. USBiological 10
Worldwide
Amitriptyline Amitriptyline is an inhibitor of serotonin reuptake transporter (SERT) and noradrenaline reuptake transporter (NET) , with K i s of 3.45 nM and 13.3 nM for human SERT and NET, respectively. Amitriptyline also weakly binds to dopamine reuptake transporter (DAT) with a K i of 2.58 μM. Amitriptyline also inhibits adrenergic , muscarinic , histamine and 5-HT receptors. Amitriptyline is a TrkA and TrkB receptors agonist with potent neurotrophic activity. Amitriptyline has antidepressant activity [1] [2] [3]. Uses: Scientific research. Group: Signaling pathways. CAS No. 50-48-6. Pack Sizes: 10 mM * 1 mL; 10 mg; 25 mg; 50 mg; 100 mg. Product ID: HY-B0527. MedChemExpress MCE
Amitriptyline-d3 hydrochloride Amitriptyline-d3 hydrochloride is the deuterium labeled Amitriptyline (hydrochloride). Amitriptyline hydrochloride is an inhibitor of serotonin reuptake transporter (SERT) and noradrenaline reuptake transporter (NET) , with K i s of 3.45 nM and 13.3 nM for human SERT and NET, respectively. Amitriptyline hydrochloride also weakly binds to dopamine reuptake transporter (DAT) with a K i of 2.58 μM. Amitriptyline hydrochloride also inhibits adrenergic , muscarinic , histamine and 5-HT receptors. Amitriptyline hydrochloride is a TrkA and TrkB receptors agonist with potent neurotrophic activity. Amitriptyline hydrochloride has antidepressant activity [1] [2] [3]. Uses: Scientific research. Group: Isotope-labeled compounds. CAS No. 342611-00-1. Pack Sizes: 5 mg; 10 mg. Product ID: HY-135096. MedChemExpress MCE
Amitriptyline hydrochloride Amitriptyline hydrochloride is an inhibitor of serotonin reuptake transporter (SERT) and noradrenaline reuptake transporter (NET) , with K i s of 3.45 nM and 13.3 nM for human SERT and NET, respectively. Amitriptyline hydrochloride also weakly binds to dopamine reuptake transporter (DAT) with a K i of 2.58 μM. Amitriptyline hydrochloride also inhibits adrenergic , muscarinic , histamine and 5-HT receptors. Amitriptyline hydrochloride is a TrkA and TrkB receptors agonist with potent neurotrophic activity. Amitriptyline hydrochloride has antidepressant activity [1] [2] [3]. Uses: Scientific research. Group: Signaling pathways. CAS No. 549-18-8. Pack Sizes: 10 mM * 1 mL; 5 g. Product ID: HY-B0527A. MedChemExpress MCE
Amitriptyline (hydrochloride) (Standard) Amitriptyline (hydrochloride) (Standard) is the analytical standard of Amitriptyline (hydrochloride). This product is intended for research and analytical applications. Amitriptyline hydrochloride is an inhibitor of serotonin reuptake transporter (SERT) and noradrenaline reuptake transporter (NET) , with K i s of 3.45 nM and 13.3 nM for human SERT and NET, respectively. Amitriptyline hydrochloride also weakly binds to dopamine reuptake transporter (DAT) with a K i of 2.58 μM. Amitriptyline hydrochloride also inhibits adrenergic , muscarinic , histamine and 5-HT receptors. Amitriptyline hydrochloride is a TrkA and TrkB receptors agonist with potent neurotrophic activity. Amitriptyline hydrochloride has antidepressant activity [1] [2] [3]. Uses: Scientific research. Group: Signaling pathways. CAS No. 549-18-8. Pack Sizes: 10 mg; 25 mg; 50 mg; 100 mg. Product ID: HY-B0527AR. MedChemExpress MCE
Apraclonidine hydrochloride Apraclonidine is an α2-adrenergic receptor (α2-AR) agonist and structural analog of clonidine. It is used for the treatment of post-surgical elevated intraocular pressure. It inhibits noradrenaline-stimulated contraction in guinea pig ileum with EC50s of 7.59 nM and rabbit vas deferens with EC50s of 6.76 nM. Uses: Adrenergic alpha-2 receptor agonists. Synonyms: ALO 2145; 2,6-Dichloro-N1-(4,5-dihydro-1H-imidazol-2-yl)-1,4-benzenediamine hydrochloride; Iopidine; p-Aminoclonidine monohydrochloride. Grades: ≥98%. CAS No. 73218-79-8. Molecular formula: C9H10Cl2N4·HCl. Mole weight: 281.6. BOC Sciences 2
ARC 239 ARC239 dihydrochloride is a potent and selective α2 B adrenoceptor antagonist. It is used as an α-adrenoceptor blocking drug. It competitively antagonizes pressor responses to adrenaline and inhibits pressor responses to noradrenaline, tyramine, phenylephrine and dimethylphenylpiperazinium. Uses: Arc239 dihydrochloride is used as an α-adrenoceptor blocking drug. Synonyms: ARC239 dihydrochloride; ARC 239 dihydrochloride; ARC-239 dihydrochloride; 2-(2-(4-(2-Methoxyphenyl)piperazin-1-yl)ethyl)-4,4-dimethyl-1,3-(2H,4H)-isoquinolindione dihydrochloride;AR-C239 Dihydrochloride. Grades: 98%. CAS No. 67339-62-2. Molecular formula: C24H29N3O3. Mole weight: 407.5. BOC Sciences 2
Atomoxetine Atomoxetine is a selective inhibitor of noradrenaline reuptake. Atomoxetine was originally called tomoxetine but changed to avoid any potential confusion with tamoxifen that might lead to errors in dispensing the drug. It is a selective norepinephrine reuptake inhibitor with Ki values of 5, 77, and 1,451 nM for norepinephrine, serotonin, and dopamine transporters, respectively. Atomoxetine (0.1, 0.5, and 1 mg/kg) reduces premature responding, a measure of impulsivity, by rats in the 5-choice serial reaction time test (5CSRTT) in a dose-dependent manner. Synonyms: N-methyl-γR-(2-methylphenoxy)-benzenepropanamine; Atomoxetine; HSDB 7352; HSDB-7352; HSDB7352. Grades: ≥98%. CAS No. 83015-26-3. Molecular formula: C17H21NO. Mole weight: 255.4. BOC Sciences
Atomoxetine hydrochloride Atomoxetine (Tomoxetine) hydrochloride is a selective noradrenaline reuptake inhibitor with K i values of 5 nM, 77 nM and 1451 nM for norepinephrine (NE), serotonin (5-HT) and dopamine (DA) transporters, respectively. Atomoxetine hydrochloride is a potent Na + channels (VGSCs) blocker. Atomoxetine hydrochloride can be used for attention-deficit hyperactivity disorder (ADHD) research [1] [2] [3]. Uses: Scientific research. Group: Signaling pathways. Alternative Names: Tomoxetine hydrochloride; (R)-Tomoxetine hydrochloride; LY 139603. CAS No. 82248-59-7. Pack Sizes: 10 mM * 1 mL; 100 mg. Product ID: HY-17385. MedChemExpress MCE
Bisindolylmaleimide VIII acetate Bisindolylmaleimide VIII (BIM VIII) is a selective protein kinase C (PKC) inhibitor with IC50 of 158 nM for rat brain that acts at the ATP binding site. Bis VIII has been previously shown to enhance Fas-mediated apoptosis through a protein kinase C-independent mechanism. BIM VIII does not inhibit the tyrosine phosphorylation or the activation of phospholipase C γ1. BIM VIII inhibits carbachol-evoked noradrenaline release from human SH-SY5Y neuroblastoma cells with an IC50 of 600 nM. Synonyms: BIM VIII; Ro 31-7549. Grades: ≥98%. CAS No. 138516-31-1. Molecular formula: C24H22N4O2·C2H4O2. Mole weight: 458.5. BOC Sciences 10
BRL 44408 Selective α2A-adrenoceptor antagonist. Increases hippocampal noradrenaline release following systemic administration. Group: Biochemicals. Alternative Names: 2-[(4,5-Dihydro-1H-imidazol-2-yl)methyl]-2,3-dihydro-1-methyl-1H-isoindole. Grades: Highly Purified. CAS No. 118343-19-4. Pack Sizes: 10mg. US Biological Life Sciences. USBiological 2
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BRL 44408 Maleate (2-[(4,5-Dihydro-1H-imidazol-2-yl)methyl]-2,3-dihydro-1-methyl-1H-isoindole Maleate) A selective alpha-2A-adrenoceptor antagonist (Ki = 1.7nM and 144.5nM at alpha-2A and alpha-2B-adrenergic receptors respectively). Has been used to study regulation of neurotransmitter release from sympathetic nerves and shown to increase hippocampal noradrenaline release following systemic administration. Group: Biochemicals. Grades: Highly Purified. CAS No. 118343-19-4. Pack Sizes: 10mg. Molecular Formula: C??H??N?; C?H?O?. US Biological Life Sciences. USBiological 4
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catechol O-methyltransferase The mammalian enzyme acts more rapidly on catecholamines such as adrenaline or noradrenaline than on catechols. Group: Enzymes. Synonyms: COMT I COMT II; S-COMT (soluble form of catechol-O-methyltransferase); MB-COMT (membrane-bound form of catechol-O-methyltransferase); catechol methyltransferase; catecholamine O-methyltransferase. Enzyme Commission Number: EC 2.1.1.6. CAS No. 9012-25-3. COMT. Storage: Store it at +4 ?C for short term. For long term storage, store it at -20 ?C?-80 ?C. Form: Liquid or lyophilized powder. EXWM-1961; catechol O-methyltransferase; EC 2.1.1.6; 9012-25-3; COMT I COMT II; S-COMT (soluble form of catechol-O-methyltransferase); MB-COMT (membrane-bound form of catechol-O-methyltransferase); catechol methyltransferase; catecholamine O-methyltransferase. Cat No: EXWM-1961. Creative Enzymes
CGP 35348 (GABAB Receptor Antagonist, CGP 35348, CGP35348, CGP-35348) A selective antagonist of post-synaptic GABAB receptors (IC50 = 34uM) that can permeate the blood brain barrier. Exhibits about 10-fold lower affinity for pre-synaptic receptors. Blocks K+-evoked glycine exocytosis in mouse spinal cord and hippocampal nerve endings. Shown to antagonize the potentiating effect of L-baclofen on noradrenaline-induced stimulation of adenylate cyclase in rat cortex slices. Group: Biochemicals. Grades: Highly Purified. CAS No. 123690-79-9. Pack Sizes: 10mg. US Biological Life Sciences. USBiological 4
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Colterol-d9 Colterol-d9 is abelled β-Adrenergic agonist and a labeled metabolite of Bitolterol. Group: Biochemicals. Alternative Names: 4-[2-[(1,1-Dimethylethyl)amino]-1-hydroxyethyl]-1,2-benzenediol-d9; (+/-)-α-[(tert-Butylamino)methyl]-3,4-dihydroxy-benzyl Alcohol-d9; (+/-)-N-t-Butylnoradrenaline-d9; (+/-)-tert-Butyl Noradrenaline-d9; dl-1-(3,4-Dihydroxyphenyl)-2-tert-butylaminoethanol-d9; dl-N-tert-Butylnorepinephrine-d9. Grades: Highly Purified. CAS No. 1346598-08-0. Pack Sizes: 1mg. US Biological Life Sciences. USBiological 2
Worldwide
Colterol Hydrochloride Colterol Hydrochloride, an impurity of Salbutamol, is used as a beta-adrenergic agonist, an anti-asthmatic drug and a bronchodilator agent. Synonyms: 4-[2-[(1,1-Dimethylethyl)amino]-1-hydroxyethyl]-1,2-benzenediol Hydrochloride; (+/-)-α-[(tert-Butylamino)methyl]-3,4-dihydroxy-benzyl Alcohol Hydrochloride; (+/-)-N-t-Butylnoradrenaline Hydrochloride; (+/-)-tert-Butyl Noradrenaline Hydrochloride; dl-1-(3,4-Dihydroxyphenyl)-2-tert-butylaminoethanol Hydrochloride; dl-N-tert-Butylnorepinephrine Hydrochloride. Grades: ≥95%. CAS No. 52872-37-4. Molecular formula: C12H20ClNO3. Mole weight: 261.74. BOC Sciences 8
Colterol Hydrochloride Colterol is β-Adrenergic agonist, and a metabolite of Bitolterol [30392-41-7]. Group: Biochemicals. Alternative Names: 4-[2-[(1,1-Dimethylethyl)amino]-1-hydroxyethyl]-1,2-benzenediol Hydrochloride; (+/-)-α-[(tert-Butylamino)methyl]-3,4-dihydroxy-benzyl Alcohol Hydrochloride; (+/-)-N-t-Butylnoradrenaline Hydrochloride; (+/-)-tert-Butyl Noradrenaline Hydrochloride; dl-1-(3,4-Dihydroxyphenyl)-2-tert-butylaminoethanol Hydrochloride; dl-N-tert-Butylnorepinephrine Hydrochloride. Grades: Highly Purified. CAS No. 52872-37-4. Pack Sizes: 25mg. US Biological Life Sciences. USBiological 2
Worldwide
Cyclopentamine Hydrochloride Cyclopentamine is a sympathomimetic alkylamine that is classified as a vasoconstrictor. Cyclopentamine is a release agent of the catecholamine neurotransmitters norepinephrine (noradrenaline), epinephrine (adrenaline), and dopamine. Synonyms: N,α-Dimethylcyclopentaneethanamine Hydrochloride; N,α-Dimethylcyclopentaneethylamine Hydrochloride; Clopane Hydrochloride; Cyclonarol Hydrochloride; Cyclopentadrin Hydrochloride; Cyclopentadrine Hydrochloride; Cyclopentamin Hydrochloride; Cyklosal Hydrochloride; Cyklosan Hydrochloride; Sinos Hydrochloride. Grades: 95%. CAS No. 538-02-3. Molecular formula: C9H20ClN. Mole weight: 177.72. BOC Sciences 8
Desmethyl Sibutramine Desmethyl Sibutramine is a metabolite of Sibutramine (S422500), a serotonin and noradrenaline reuptake inhibitor (SNR). Decreases calorie intake and increases energy expenditure. Group: Biochemicals. Grades: Highly Purified. CAS No. 168835-59-4. Pack Sizes: 5mg, 50mg. Molecular Formula: C16H24ClN. US Biological Life Sciences. USBiological 2
Worldwide
Desmethyl Sibutramine-d6, Hydrochloride A labeled metabolite of Sibutramine, a serotonin and noradrenaline reuptake inhibitor (SNR). Decreases calorie intake and increases energy expenditure. Group: Biochemicals. Grades: Highly Purified. Pack Sizes: 1mg. US Biological Life Sciences. USBiological 1
Worldwide
Desmethyl Sibutramine, Hydrochloride Salt A metabolite of Sibutramine, a serotonin and noradrenaline reuptake inhibitor (SNR). Decreases calorie intake and increases energy expenditure. Group: Biochemicals. Alternative Names: 1-(4-Chlorophenyl)-N-methyl-α-(2-methylpropyl)-cyclobutanemethanamine Hydrochloride. Grades: Highly Purified. CAS No. 84467-94-7. Pack Sizes: 5mg. US Biological Life Sciences. USBiological 3
Worldwide
Diclofensine Diclofensine is a potent inhibitor of monoamine reuptake, blocking the uptake of dopamine (IC50=0.74 nM), as an effective antidepressant. Uses: A stimulant; inhibits reuptake of dopamine and noradrenaline, is an effective antidepressant. compound exhibits significant addictive properties. Synonyms: 4-(3,4-Dichlorophenyl)-1,2,3,4-tetrahydro-7-methoxy-2-methyl-isoquinoline; Ro 8-4650; 4-(3,4-dichlorophenyl)-7-methoxy-2-methyl-1,2,3,4-tetrahydroisoquinoline. Grades: ≥98%. CAS No. 67165-56-4. Molecular formula: C17H17Cl2NO. Mole weight: 322.23. BOC Sciences 11
Diclofensine-d3 Hydrochloride Labeled Diclofensine. Diclofensine is a stimulant; inhibits reuptake of dopamine and noradrenaline, is an effective antidepressant. Diclofensine exhibits significant addictive properties. Group: Biochemicals. Alternative Names: 4-(3,4-Dichlorophenyl)-1,2,3,4-tetrahydro-7-methoxy-2-(methyl)isoquinoline Hydrochloride. Grades: Highly Purified. Pack Sizes: 1mg. US Biological Life Sciences. USBiological 2
Worldwide
Diclofensine (hydrochloride) Diclofensine inhibits reuptake of dopamine and noradrenaline with IC50 values of 0.74, 2.3, and 3.7 nM, respectively. Uses: Diclofensine inhibits reuptake of dopamine and noradrenaline. Synonyms: Diclofensine HCl; Moxifensine hydrochloride; Ro-84650; Moxifensine HCl; Ro 84650; Ro84650; Diclofensine Hydrochloride; 4-(3,?4-dichlorophenyl)?-1,?2,?3,?4-tetrahydro-7-methoxy-2-methyl-isoquinoline, monohydrochloride. Grades: ≥98%. CAS No. 34041-84-4. Molecular formula: C17H17Cl2NO HCl. Mole weight: 358.7. BOC Sciences 11
Diclofensine Hydrochloride Diclofensine is a stimulant; inhibits reuptake of dopamine and noradrenaline, is an effective antidepressant. Diclofensine exhibits significant addictive properties. Group: Biochemicals. Alternative Names: 4-(3,4-Dichlorophenyl)-1,2,3,4-tetrahydro-7-methoxy-2-methylisoquinoline Hydrochloride. Grades: Highly Purified. CAS No. 34041-84-4. Pack Sizes: 10mg. US Biological Life Sciences. USBiological 2
Worldwide
Didesmethyl Sibutramine A metabolite of Sibutramine, a serotonin and noradrenaline reuptake inhibitor (SNR). Decreases calorie intake and increases energy expenditure. Group: Biochemicals. Grades: Highly Purified. Pack Sizes: 5mg. US Biological Life Sciences. USBiological 1
Worldwide
Didesmethyl Sibutramine-d6 A labeled metabolite of Sibutramine, a serotonin and noradrenaline reuptake inhibitor (SNR). Decreases calorie intake and increases energy expenditure. Group: Biochemicals. Grades: Highly Purified. Pack Sizes: 1mg. US Biological Life Sciences. USBiological 1
Worldwide
D,L N,O-Didesmethylvenlafaxine A metabolite of Venlafaxine, a selective serotonin noradrenaline reuptake inhibitor. Group: Biochemicals. Grades: Highly Purified. Pack Sizes: 5mg. US Biological Life Sciences. USBiological 1
Worldwide
DL-Norepinephrine Hydrochloride Norepinephrine is the neurotransmitter at most sympathetic neuroeffector junctions and has pharmacologic activities on both α1 and β1 adrenoceptors. Uses: Adrenergic alpha-agonists. Synonyms: 4-(2-Amino-1-hydroxyethyl)-1,2-benzenediol; (+/-)-Noradrenaline Hydrochloride; DL-Arterenol Hydrochloride; NSC 7930; dl-Noradrenaline Hydrochloride; dl-Norepinephrine Hydrochloride. Grades: ≥95%. CAS No. 55-27-6. Molecular formula: C8H12ClNO3. Mole weight: 205.64. BOC Sciences 8
DL-Normetanephrine Glucuronide A derivative of Norepinephrine. Norepinephrine, also known as noradrenaline, is a marker for catecholamine-secreting tumors such as pheochromocytoma, paraganglioma, and neuroblastoma. Synonyms: 4-(2-amino-1-hydroxyethyl)benzene-1,2-diol Glucuronide. Grades: > 95%. Molecular formula: C15H21NO9. Mole weight: 359.34. BOC Sciences 8
D,L-O-Desmethylvenlafaxine (4-[2-(Dimethylamino)-1-(1-hydroxycyclo-hexyl)ethyl]phenol) A metabolite of Venlafaxine, a selective serotonin noradrenaline reuptake inhibitor. Used as an antidepressant. Group: Biochemicals. Alternative Names: 4-[2-(Dimethylamino)-1-(1-hydroxycyclo-hexyl)ethyl]phenol. Grades: Highly Purified. Pack Sizes: 5mg. US Biological Life Sciences. USBiological 1
Worldwide
D,L-O-Desmethylvenlafaxine-d6 (4-[2-(Dimethylamino)-1-(1-hydroxycyclo-hexyl)ethyl]phenol-d6) A deuterated metabolite of Venlafaxine, a selective serotonin noradrenaline reuptake inhibitor. Used as an antidepressant. Group: Biochemicals. Alternative Names: 4-[2-(Dimethylamino)-1-(1-hydroxycyclo-hexyl)ethyl]phenol-d6. Grades: Highly Purified. CAS No. Unlabeled: 93413-62-8 Labeled: 1020719-35-0. Pack Sizes: 1mg, 10mg. Molecular Formula: C??H??D?NO?, Molecular Weight: 269.41. US Biological Life Sciences. USBiological 1
Worldwide
D,L-Venlafaxine (1-[2- (Dimethylamino) -1- (4-methoxyphenyl) ethyl]cyclohexanol) A selective serotonin noradrenaline reuptake inhibitor. Used as an antidepressant. Group: Biochemicals. Alternative Names: 1-[2- (Dimethylamino) -1- (4-methoxyphenyl) ethyl]cyclohexanol. Grades: Highly Purified. Pack Sizes: 50mg. US Biological Life Sciences. USBiological 1
Worldwide
D,L-Venlafaxine-d6 (1-[2- (Dimethylamino) -1- (4-methoxyphenyl) ethyl]cyclohexanol-d6) Labelled Venlafaxine, a selective serotonin noradrenaline reuptake inhibitor. Venlafaxine is used as an antidepressant. Group: Biochemicals. Alternative Names: 1-[2- (Dimethylamino) -1- (4-methoxyphenyl) ethyl]cyclohexanol-d6. Grades: Highly Purified. Pack Sizes: 5mg. US Biological Life Sciences. USBiological 1
Worldwide
D,L-Venlafaxine, Hydrochloride (1-[2- (Dimethylamino) -1- (4-methoxyphenyl) ethyl]cyclohexanol, HCl) A selective serotonin noradrenaline reuptake inhibitor. Used as an antidepressant. Group: Biochemicals. Alternative Names: 1-[2- (Dimethylamino) -1- (4-methoxyphenyl) ethyl]cyclohexanol, HCl. Grades: Highly Purified. CAS No. 99300-78-4. Pack Sizes: 100mg. US Biological Life Sciences. USBiological 1
Worldwide
Dothiepin Dothiepin (Dosulepin; Dothep) is an antidepressant agent with sedative/anxiolytic activity. Dothiepin is an inhibitor preferring of noradrenaline uptake than serotonin uptake. Dothiepin facilitates noradrenergic neurotransmission via inhibiting the neuronal uptake. Dothiepin is also an antagonist of histamine H1-receptor without cardiotoxicity. Dothiepin exhibits significant analgesic activity in psychogenic facial pain, idiopathic fibromyalgia syndrome or rheumatoid arthritis [1]. Uses: Scientific research. Group: Signaling pathways. Alternative Names: Dosulepin; Dothep. CAS No. 113-53-1. Pack Sizes: 1 mg. Product ID: HY-12394. MedChemExpress MCE
Droxidopa Droxidopa is a synthetic amino acid precursor which acts as a prodrug to the neurotransmitters norepinephrine (noradrenaline) and epinephrine (adrenaline). It is capable of crossing the protective blood-brain barrier. Synonyms: (βR)-β,3-Dihydroxy-L-tyrosine; threo-β,3-Dihydroxy-L-tyrosine; L-threo-3-(3,4-Dihydroxyphenyl)serine; (-)-threo-3,4-Dihydroxyphenylserine; (2S,3R)-3-(3,4-Dihydroxyphenyl)-2-amino-3-hydroxypropanoic Acid; DOPS; L-DOPS; L-Threodops; L-threo-3,4-Dihydroxyphenylserine; L-threo-DOPS; L-threo-β-(3,4-Dihydroxyphenyl)serine; SM 5688; threo-Dopaserine. Grades: >98%. CAS No. 23651-95-8. Molecular formula: C9H11NO5. Mole weight: 213.19. BOC Sciences
Erythro-β,3-dihydroxy-DL-tyrosine Erythro-β,3-dihydroxy-DL-tyrosine is an impurity of Droxidopa, which is a synthetic amino acid precursor used as a prodrug to the neurotransmitter norepinephrine (noradrenaline). Synonyms: Droxidopa Impurity 11 (DL-erythro-Droxidopa); DL-erythro-3,4-Dihydroxyphenylserine; Erythro-2-Amino-3-(3,4-dihydroxyphenyl)-3-hydroxypropionic Acid; Erythro-3-(3,4-Dihydroxyphenyl)serine; rel-(βR)-β,3-Dihydroxy-D-tyrosine; DL-Tyrosine, β,3-dihydroxy-, erythro-; Serine, 3-(3,4-dihydroxyphenyl)-, DL-erythro-; D-Tyrosine, β,3-dihydroxy-, (βR)-rel-. CAS No. 16322-99-9. Molecular formula: C9H11NO5. Mole weight: 213.19. BOC Sciences 8
Guanoclor Guanoclor is an antihypertensive compound. Guanoclor is an adrenergic neurone-blocking agent, which also interferes with noradrenaline synthesis by inhibition of the enzyme dopamine beta-hydroxylase [1]. Uses: Scientific research. Group: Signaling pathways. Alternative Names: Vatensol. CAS No. 5001-32-1. Pack Sizes: 5 mg; 10 mg; 25 mg; 50 mg; 100 mg. Product ID: HY-100796. MedChemExpress MCE

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