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1,2,3,4,5,6-Benzenehexamine trihydrochloride is used as a reagent in the preparation of 2-(benzimidazol-2-yl)quinoxalines as selective antagonists at human A1 and A3 adenosine receptors. Group: Biochemicals. Grades: Highly Purified. CAS No. 126521-82-2. Pack Sizes: 25mg, 50mg. Molecular Formula: C6H15Cl3N6. US Biological Life Sciences.
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1,2,3,4,5,6-Benzenehexamine Trihydrochloride
1,2,3,4,5,6-Benzenehexamine Trihydrochloride. Uses: Designed for use in research and industrial production. Additional or Alternative Names: Benzene-1,2,3,4,5,6-hexaamine trihydrochloride. Product Category: Other Monomers. CAS No. 126521-82-2. Molecular formula: C6H12N6·3HCl. Mole weight: 204.66 g/mol. Purity: 0.97. Product ID: ACM-MO-126521822. Alfa Chemistry ISO 9001:2015 Certified.
1,3,5-Triaminobenzene trihydrochloride
1,3,5-Triaminobenzene trihydrochloride. Group: Biochemicals. Grades: Highly Purified. CAS No. 638-09-5,108-72-5. Pack Sizes: 2g, 5g, 10g, 25g, 50g. Molecular Formula: C6H12Cl3N3. US Biological Life Sciences.
(-)-15-Deoxyspergualin trihydrochloride is an antineoplastic agent. Synonyms: Gusperimus (-)-form trihydrochloride; (-)-Gusperimus trihydrochloride. Grade: 95%. CAS No. 84937-45-1. Molecular formula: C17H40Cl3N7O3. Mole weight: 496.904.
(-)-15-Deoxyspergualin Trihydrochloride
(-)-15-Deoxyspergualin Trihydrochloride is an immunosuppressive drug with potential use in the treatment of transplant rejection. Group: Biochemicals. Grades: Highly Purified. CAS No. 84937-45-1. Pack Sizes: 1mg, 10mg. Molecular Formula: C17H40Cl3N7O3, Molecular Weight: 496.9. US Biological Life Sciences.
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1-Naphthylacetyl Spermine Trihydrochloride
A poliamine amide as potent Spermidine uptake inhibitor. Group: Biochemicals. Alternative Names: N- [3- [ [4- [ (3-Aminopropyl) amino] butyl] amino] propyl] -1-naphthaleneacetamide Trihydrochloride. Grades: Highly Purified. CAS No. 1049731-36-3. Pack Sizes: 25mg. US Biological Life Sciences.
An impurity of Plerixafor which is an antagonist of the CXCR4 chemokine receptor. Synonyms: Plerixafor Impurity 08. CAS No. 128495-30-7. Molecular formula: C17H31ClN4O2S. Mole weight: 390.97.
2-[5-Chloro-2-[[3- (4-methylpiperazin-1-yl) propyl]amino]pyrimidin-4-yl]benzo[b]thiophene-4-carboxamide N-cyclopropyl Trihydrochloride is an inhibitor of IkB-kinase (IKK2). Small molecules that inhibits IkB-kinase and NF-κB pathways are potential anti-inflammatory drug candidate. Group: Biochemicals. Grades: Highly Purified. CAS No. 946518-60-1. Pack Sizes: 1mg, 2.5mg. Molecular Formula: C24H32Cl4N6OS, Molecular Weight: 594.429999999999. US Biological Life Sciences.
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2-Pyridin-3-Yl Piperazine Trihydrochloride
2-Pyridin-3-Yl Piperazine Trihydrochloride. Group: Biochemicals. Grades: Highly Purified. Pack Sizes: 50mg, 100mg, 250mg, 500mg, 1g. US Biological Life Sciences.
3- [ [3- [ (4-Aminobutyl) amino] propyl] amino] propanenitrile Trihydrochloride is an intermediate in the synthesis of Thermospermine (T343890), a structure isomer of Spermine (S680510). Group: Biochemicals. Grades: Highly Purified. Pack Sizes: 25mg, 100mg. Molecular Formula: C10H25Cl3N4. US Biological Life Sciences.
3-[4-(4-Methoxyphenyl)piperazinyl]azetidine trihydrochloride. Uses: Designed for use in research and industrial production. Additional or Alternative Names: 3-[4-(4-Methoxyphenyl)piperazinyl]azetidine trihydrochloride;1-AZETIDIN-3-YL-4-(4-METHOXY-PHENYL)-PIPERAZINE TRIHYDROCHLORIDE;3-4-(4-METHOXYPHENYL)PIPERAZINYLAZETIDINE 3HCL;3-(4-(p-methoxyphenyl)piperazinyl)azetidinetrihydrochloride;3-(4-(O-METHOXYPHENYL. Product Category: Heterocyclic Organic Compound. CAS No. 223381-99-5. Molecular formula: C14H21N3O.3(HCl). Mole weight: 356.72. Purity: 0.96. IUPACName: 1-(azetidin-3-yl)-4-(4-methoxyphenyl)piperazine;trihydrochloride. Canonical SMILES: COC1=CC=C(C=C1)N2CCN(CC2)C3CNC3.Cl.Cl.Cl. Product ID: ACM223381995. Alfa Chemistry ISO 9001:2015 Certified.
3-[4-(4-Tolyl)piperazinyl]azetidine trihydrochloride. Uses: Designed for use in research and industrial production. Additional or Alternative Names: 3-[4-(4-Tolyl)piperazinyl]azetidine trihydrochloride;3-4-(4-TOLYL)PIPERAZINYLAZETIDINE 3HCL;3-(4-(P-METHYLPHENYL)PIPERAZINYL)AZETIDINE TRIHYDROCHLORIDE. Product Category: Heterocyclic Organic Compound. CAS No. 223382-00-1. Molecular formula: C14H24Cl3N3. Mole weight: 340.71946. Purity: 0.96. IUPACName: tert-butyl 6-hydroxy-2-[(2-methylpropan-2-yl)oxycarbonylamino]hexanoate. Canonical SMILES: CC1=CC=C(C=C1)N2CCN(CC2)C3CNC3.Cl.Cl.Cl. Product ID: ACM223382001. Alfa Chemistry ISO 9001:2015 Certified.
4-(2-Morpholinoethoxy)benzene-1,2-diamine trihydrochloride. Uses: Designed for use in research and industrial production. Additional or Alternative Names: 4-(2-Morpholinoethoxy)benzene-1,2-diamine trihydrochloride, 75328-29-9, RP07027, Y4003. Product Category: Heterocyclic Organic Compound. CAS No. 75328-29-9. Molecular formula: C12H19N3O2·3HCl. Mole weight: 346.68. Purity: 0.96. IUPACName: 4-(2-morpholin-4-ylethoxy)benzene-1,2-diamine;trihydrochloride. Canonical SMILES: C1COCCN1CCOC2=CC(=C(C=C2)N)N.Cl.Cl.Cl. Product ID: ACM75328299. Alfa Chemistry ISO 9001:2015 Certified.
4-[5-(4-Methyl-1-piperazinyl)-1H,1'H-2,5'-bibenzimidazol-2'-yl]phenol trihydrochloride. Group: Biochemicals. Alternative Names: Hoechst 33258; bisBenzimide H33258. Grades: Highly Purified. CAS No. 23491-45-4. Pack Sizes: 25mg, 50mg, 100mg, 250mg, 500mg. Molecular Formula: C25H24N6O·3HCl. US Biological Life Sciences.
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A 419259 trihydrochloride
A 419259 trihydrochloride. Group: Biochemicals. Grades: Purified. CAS No. 1435934-25-0. Pack Sizes: 10mg. US Biological Life Sciences.
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A 419259 trihydrochloride
A 419259 trihydrochloride is a Src family kinases inhibitor with IC50s of 9 nM, 3 nM and 3 nM for Src, Lck and Lyn, respectively[1][2]. Uses: Scientific research. Group: Signaling pathways. Alternative Names: RK 20449 trihydrochloride. CAS No. 1435934-25-0. Pack Sizes: 5 mg; 10 mg; 50 mg; 100 mg. Product ID: HY-15764A.
A 419259 trihydrochloride
Potent Hck inhibitor (IC50 = 0.43 nM). Also inhibits other Src family kinases (SFKs). Suppresses proliferation and induces apoptosis in CML cell lines including CD34+. Also inhibits acute myeloid leukemia (AML) stem cell proliferation in vitro and in vivo. Synonyms: A419259 trihydrochloride; A-419259 trihydrochloride; RK 20449 trihydrochloride; RK20449 trihydrochloride; RK-20449 trihydrochloride. Grade: >98%. CAS No. 1435934-25-0. Molecular formula: C29H37Cl3N6O. Mole weight: 592.0.
ABT 724 trihydrochloride. Group: Biochemicals. Grades: Purified. CAS No. 587870-77-7. Pack Sizes: 10mg, 50mg. US Biological Life Sciences.
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Arg-Arg β-Naphthylamide Trihydrochloride
A specific substrate for dipeptidyl peptidase III. Synonyms: Arg-Arg beta-naphthylamide trihydrochloride; H-Arg-Arg-βNA 3 HCl; L-Argininamide,L-arginyl-N-2-naphthalenyl-, trihydrochloride (9CI). Grade: 95%. CAS No. 100900-26-3. Molecular formula: C22H36Cl3N9O2. Mole weight: 564.94.
Atazanavir Hydrazine Analog Trihydrochloride
An intermediate for the synthesis of Atazanavir and the preparation of some peptide analogs. Synonyms: Des-N-(methoxycarbonyl)-L-tert-leucine Atazanavir Trihydrochloride. Grade: > 95%. CAS No. 198904-87-9. Molecular formula: C22H26N4O. 3 HCl. Mole weight: 362.48 3 36.46.
ATM-3507 trihydrochloride
ATM-3507 is an inhibitor of tropomyosin. In human melanoma cell lines, the IC50s are 3.83-6.84 μM. Grade: 98%. Molecular formula: C37H49Cl3FN5O2. Mole weight: 721.17.
Avotaciclib trihydrochloride
Avotaciclib trihydrochloride is a potent and orally active CDK1 inhibitor that can be studied in locally advanced or metastatic pancreatic cancer. Synonyms: BEY1107 trihydrochloride; 3-Pyridinol, 2,6-bis(2-amino-4-pyrimidinyl)-, hydrochloride (1:3). CAS No. 1983984-01-5. Molecular formula: C13H11N7O.3HCl. Mole weight: 390.66.
AXC-715 trihydrochloride
AXC-715 trihydrochloride is a dual agonist of TLR7/TLR8. (Extracted from patent WO2020168017 A1). Synonyms: 1-(4-Aminobutyl)-2-butyl-1H-imidazo[4,5-c]quinolin-4-amine Trihydrochloride; 1H-Imidazo[4,5-c]quinoline-1-butanamine, 4-amino-2-butyl-, hydrochloride (1:3). Grade: 95%. CAS No. 2479276-17-8. Molecular formula: C18H28Cl3N5. Mole weight: 420.81.
BI-9321 trihydrochloride
BI-9321 trihydrochloride is a potent, selective and cellular active nuclear receptor-binding SET domain 3 (NSD3)-PWWP1 domain antagonist with a Kd value of 166 nM. BI-9321 trihydrochloride is inactive against NSD2-PWWP1 and NSD3-PWWP2. BI-9321 trihydrochloride specifically disrupts histone interactions of the NSD3-PWWP1 domain with an IC50 of 1.2 ?M in U2OS cells[1]. Uses: Scientific research. Group: Signaling pathways. CAS No. 2387510-87-2. Pack Sizes: 10 mM * 1 mL; 5 mg; 10 mg; 25 mg; 50 mg; 100 mg. Product ID: HY-114208A.
Bisbenzimide H 33258 Fluorochrome, Trihydrochloride - CAS 23491-45-4
for fluorescence, ?97.0% (HPLC). Group: Fluorescence/luminescence spectroscopy.
BIX 01294 trihydrochloride
BIX 01294 is a G9a histone methyltransferase inhibitor. It enhances the induction of pluripotent stem cells from somatic cells in vitro. BIX-01294 trihydrochloride induces necroptosis and autophagy. Synonyms: BIX 01294 trihydrochloride; BIX-01294; N-(1-benzylpiperidin-4-yl)-6,7-dimethoxy-2-(4-methyl-1,4-diazepan-1-yl)quinazolin-4-amine trihydrochloride. Grade: >98%. CAS No. 1392399-03-9. Molecular formula: C28H41Cl3N6O2. Mole weight: 600.02.
BIX 01294 Trihydrochloride
G9a-like protein and G9a histone lysine methyltransferase (HMTase) inhibitor that H3K9me2 chromatin levels modulates H3K9me2 levels in mammalian cells and potentiates induction of pluripotent stem cells from somatic cells in vitro. Group: Biochemicals. Alternative Names: 2-(Hexahydro-4-methyl-1H-1,4-diazepin-1-yl)-6,7-dimethoxy-N-[1-(phenylmethyl)-4-piperidinyl]-4-quinazolinamine Trihydrochloride. Grades: Highly Purified. Pack Sizes: 25mg. US Biological Life Sciences.
Braco-19 trihydrochloride is a potent telomerase/telomere inhibitor, preventing the capping and catalytic action of telomerase. Braco-19 acts as G-quadruplex (GQ) binding ligand, stabilizing G-quadruplexes formation at the 3V telomeric DNA overhang and produce rapid senescence or selective cell death. Braco-19 is also a HAdV virus replication inhibitor[1][2]. Uses: Scientific research. Group: Signaling pathways. CAS No. 1177798-88-7. Pack Sizes: 10 mM * 1 mL; 5 mg; 10 mg; 25 mg; 50 mg; 100 mg. Product ID: HY-15523A.
BRACO 19 trihydrochloride
BRACO 19 trihydrochloride is a telomerase inhibitor (IC50 = 115 nM) that suppresses the expression of human telomerase reverse transcriptase (hTERT) and induces cellular senescence. BRACO 19 was shown to inhibit growth of uterine cancer cells in vitro and growth of uterine tumor xenografts in mice. Synonyms: N,N'-[9[[4-(Dimethylamino)phenyl]amino]-3,6-acridinediyl]bis-1-pyrrolidinepropanamide trihydrochloride. Grade: ≥95% by HPLC. CAS No. 1177798-88-7. Molecular formula: C35H43N7O2.3HCl. Mole weight: 703.14.
CBB1007 trihydrochloride
CBB1007 trihydrochloride, a cell-permeable amidino-guanidinium compound, is a potent, reversible and substrate competitive LSD1 selective inhibitor with an IC50 of 5.27 μM for hLSD1. Synonyms: Methyl 3-{[4-(4-carbamimidoylbenzoyl)-1-piperazinyl]carbonyl}-5-[(4-carbamimidoyl-1-piperazinyl)methyl]benzoate trihydrochloride; Benzoic acid, 3-[[4-[4-(aminoiminomethyl)benzoyl]-1-piperazinyl]carbonyl]-5-[[4-(aminoiminomethyl)-1-piperazinyl]methyl]-, methyl ester, hydrochloride (1:3). Grade: ≥96%. Molecular formula: C27H37Cl3N8O4. Mole weight: 643.99.
CHIR 99021 trihydrochloride
CHIR 99021 is a highly selective GSK-3 inhibitor. CHIR 99021 is used in the treatment of parkinsonism. Uses: The treatment of parkinsonism. Synonyms: CHIR-99021 trihydrochloride; CHIR 99021 trihydrochloride; CHIR99021 trihydrochloride; 6-[[2-[[4-(2,4-Dichlorophenyl)-5-(5-methyl-1H-imidazol-2-yl)-2-pyrimidinyl]amino]ethyl]amino]-3-pyridinecarbonitrile trihydrochloride. Grade: ≥98% by HPLC. CAS No. 1782235-14-6. Molecular formula: C22H18Cl2N8.3HCl. Mole weight: 574.72.
CHIR 99021 trihydrochloride
CHIR 99021 trihydrochloride. Group: Biochemicals. Grades: Purified. Pack Sizes: 10mg, 50mg. US Biological Life Sciences.
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Chlorhexidine Digluconate Trihydrochloride Impurity N
Chlorhexidine Digluconate Impurity N Trihydrochloride is a degradation product found in chlorhexidine digluconate solution. Group: Biochemicals. Alternative Names: N-[6-[ (Aminoiminomethyl) amino]hexyl]-N'- (4-chlorophenyl) -imidodicarbonimidic diamide Trihydrochloride. Grades: Highly Purified. Pack Sizes: 25mg. US Biological Life Sciences.
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CI 898 trihydrochloride
CI 898 trihydrochloride. Group: Biochemicals. Grades: Purified. CAS No. 82952-64-5. Pack Sizes: 10mg. US Biological Life Sciences.
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CM-579 trihydrochloride
CM-579 trihydrochloride is a first-in-class reversible and dual inhibitor of G9a and DNMT, with IC50s of 16 nM and 32 nM, respectively. It has potent in vitro cellular activity in a wide range of cancer cells. Synonyms: 6-Methoxy-2-(5-methyl-2-furyl)-N-[(1-methyl-4-piperidinyl)methyl]-7-[3-(1-pyrrolidinyl)propoxy]-4-quinolinamine trihydrochloride; 4-Quinolinamine, 6-methoxy-2-(5-methyl-2-furanyl)-N-[(1-methyl-4-piperidinyl)methyl]-7-[3-(1-pyrrolidinyl)propoxy]-, hydrochloride (1:3). Grade: ≥95%. Molecular formula: C29H43Cl3N4O3. Mole weight: 602.04.
DDP-38003 trihydrochloride
DDP-38003 trihydrochloride is the trihydrochloride salt of DDP-38003 which is a potent, selective, oral bioavailable irreversible inhibitor of KDM1A. Synonyms: DDP-38003 trihydrochloride; DDP 38003 trihydrochloride; DDP38003 trihydrochloride; N-[4-[(1S,2R)-2-aminocyclopropyl]phenyl]-4-(4-methylpiperazin-1-yl)benzamide; trihydrochloride; DDP-38003 (trihydrochloride). Molecular formula: C21H29Cl3N4O. Mole weight: 459.84.
Desmethyl-WAY 100635 trihydrochloride is a precursor for labeling the 5-HT1A antagonist WAY 100635 and can be used for PET radioligand. Synonyms: DWAY; Cyclohexanecarboxylic acid {2-[4-(2-hydroxy-phenyl)-piperazin-1-yl]-ethyl}-pyridin-2-yl-amide trihydrochloride. Grade: 98%. CAS No. 2108805-94-1. Molecular formula: C24H32N4O2.3HCl. Mole weight: 517.92.
An intermediate for the synthesis of Atazanavir. Group: Biochemicals. Alternative Names: (αS, βS)- β -Amino-α - [ [1- [ [4- (2-pyridinyl) phenyl] methyl] hydrazino] methyl] benzenepropanol Trihydrochloride; [S-(R*,R*)]- β -Amino-α - [ [1- [ [4- (2-pyridinyl) phenyl] methyl] hydrazino] methyl] benzenepropanol Trihydrochloride. Grades: Highly Purified. CAS No. 198904-87-9. Pack Sizes: 5mg. US Biological Life Sciences.
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diABZI STING agonist 1 trihydrochloride
diABZI STING agonist-1-trihydrochloride is an agonist of stimulator of interferon genes (STING) for treating cancer. Synonyms: 1H-Benzimidazole-5-carboxamide, 1-[(2E)-4-[5-(aminocarbonyl)-2-[[(1-ethyl-3-methyl-1H-pyrazol-5-yl)carbonyl]amino]-7-methoxy-1H-benzimidazol-1-yl]-2-buten-1-yl]-2-[[(1-ethyl-3-methyl-1H-pyrazol-5-yl)carbonyl]amino]-7-[3-(4-morpholinyl)propoxy]-, hydrochloride (1:3); (E)-1-(4-(5-Carbamoyl-2-(1-ethyl-3-methyl-1H-pyrazole-5-carboxamido)-7-(3-morpholinopropoxy)-1H-benzo[d]imidazol-1-yl)but-2-en-1-yl)-2-(1-ethyl-3-methyl-1H-pyrazole-5-carboxamido)-7-methoxy-1H-benzimidazole-5-carboxamide tris(hydrochloride); DiABZI. Grade: ≥98%. CAS No. 2138299-34-8. Molecular formula: C42H54Cl3N13O7. Mole weight: 959.32.
diABZI STING agonist-1 trihydrochloride
diABZI STING agonist-1 (trihydrochloride) is a selective stimulator of interferon genes (STING) receptor agonist, with EC50s of 130, 186 nM for human and mouse, respectively. Uses: Scientific research. Group: Signaling pathways. CAS No. 2138299-34-8. Pack Sizes: 10 mM * 1 mL; 1 mg; 5 mg; 10 mg; 25 mg; 50 mg; 100 mg. Product ID: HY-112921B.
GR 144053 trihydrochloride
GR 144053 trihydrochloride. Group: Biochemicals. Grades: Purified. CAS No. 1215333-48-4. Pack Sizes: 10mg, 50mg. US Biological Life Sciences.
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GR 144053 trihydrochloride
GR 144053 trihydrochloride is a potent and selective orally bioactive platelet fibrinogen receptor glycoprotein IIb/IIIa (GpIIb/IIIa) antagonist (IC50 = 37 nM). GR 144053 potently inhibits thrombus formation in vivo. Synonyms: GR 144053; GR-144053; GR144053; GR 144053 trihydrochloride. 4-[4-[4-(Aminoiminomethyl)phenyl]-1-piperazinyl]-1-piperidineacetic acid trihydrochloride. Grade: ≥99% by HPLC. CAS No. 1215333-48-4. Molecular formula: C18H27N5O2.3HCl. Mole weight: 454.83.
Gusperimus trihydrochloride
Gusperimus is a derivative of the anti-tumor antibiotic spergualin, which has immunosuppressive activity. Synonyms: Spanidin; NKT-01. Grade: 98%. CAS No. 85468-01-5. Molecular formula: C17H37N7O3.3HCl. Mole weight: 496.91.
Gusperimus Trihydrochloride
Gusperimus Trihydrochloride is an immunosuppressive agent, which was effective both in preventing and treating graft-vs.-host disease in mice. Group: Biochemicals. Grades: Highly Purified. CAS No. 85468-01-5. Pack Sizes: 1mg, 2.5mg. Molecular Formula: C17H37N7O3; 3(HCl), Molecular Weight: 387.523364599999. US Biological Life Sciences.
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GW 791343 trihydrochloride
GW791343 HCl is aHCl salt form of GW791343, which is a non-competitive allosteric modulator of human P2X7 receptor inhibitor with pIC50 of 7. Synonyms: GW791343; GW 791343; GW-791343; 1019779-04-4. Grade: >98%. CAS No. 309712-55-8. Molecular formula: C20H24F2N4O.3HCl. Mole weight: 483.81.
GW 791343 Trihydrochloride
GW 791343 Trihydrochloride. Group: Biochemicals. Alternative Names: 2-[ (3, 4-Difluorophenyl) amino]-N-[2-methyl-5- (1-piperazinylmethyl) phenyl]acetamide Trihydrochloride. Grades: Highly Purified. CAS No. 1019779-04-4. Pack Sizes: 10mg. Molecular Formula: C20H27Cl3F2N4O, Molecular Weight: 447.35. US Biological Life Sciences.
Worldwide
HM03 trihydrochloride
HM03 trihydrochloride is a potent and selective inhibitor of HSPA5 (Heat shock 70kDa protein 5, also known as Bip, Grp78) with anticancer activity. Synonyms: 4-[(6-Chloro-2-methoxy-9-acridinyl)amino]-2-[(4-methyl-1-piperazinyl)methyl]phenol trihydrochloride; Phenol, 4-[(6-chloro-2-methoxy-9-acridinyl)amino]-2-[(4-methyl-1-piperazinyl)methyl]-, hydrochloride (1:3). Grade: ≥95%. CAS No. 1082532-95-3. Molecular formula: C26H30Cl4N4O2. Mole weight: 572.35.
Hoechst 33342 trihydrochloride
Hoechst 33342 trihydrochloride is a marker dye in Hoechst series. Hoechst is A live nuclear marker dye. Hoechst binds to the grooves in the DNA double strand, which tends to be A/ T-rich DNA strand. Although it binds to all nucleic acids, the A/ T-rich double strand DNA significantly enhances fluorescence intensity Therefore,Hoechst dye can be used for living cell labeling. The fluorescence intensity of Hoechst dye increases with the increase of pH of solution[1]. Uses: Scientific research. Group: Fluorescent dye. Alternative Names: bisBenzimide H 33342 trihydrochloride; HOE 33342 trihydrochloride. CAS No. 875756-97-1. Pack Sizes: 50 mg; 100 mg. Product ID: HY-15559A.
Selective D4 receptor antagonist with excellent brain penetration. Displays an affinity (Ki) of 0.4nM for human D4 receptors with >1000-fold binding selectivity over D2 and D3 receptors. Does not block agonist-induced activation of GIRK currents. It is used frequently in retinal and CNS studies of D4 modulation. Group: Biochemicals. Grades: Highly Purified. CAS No. 158985-00-3. Pack Sizes: 10mg. US Biological Life Sciences.
Laduviglusib (CHIR-99021) trihydrochloride is a potent and selective GSK-3?/? inhibitor with IC50s of 10 nM and 6.7 nM. Laduviglusib trihydrochloride shows >500-fold selectivity for GSK-3 over CDC2, ERK2 and other protein kinases. Laduviglusib trihydrochloride is also a potent Wnt/?-catenin signaling pathway activator. Laduviglusib trihydrochloride enhances mouse and human embryonic stem cells self-renewal. Laduviglusib trihydrochloride induces autophagy[1][2][3]. Uses: Scientific research. Group: Signaling pathways. Alternative Names: CHIR-99021 trihydrochloride; CT99021 trihydrochloride. CAS No. 1782235-14-6. Pack Sizes: 10 mM * 1 mL; 5 mg; 10 mg; 25 mg; 50 mg; 100 mg. Product ID: HY-10182B.
Mavorixafor trihydrochloride (AMD-070 trihydrochloride) is a potent, selective and orally available CXCR4 antagonist, with an IC50 value of 13 nM against CXCR4 125I-SDF binding, and also inhibits the replication of T-tropic HIV-1 (NL4.3 strain) in MT-4 cells and PBMCs with an IC50 of 1 and 9 nM, respectively.Mavorixafor trihydrochloride can be used for the study of WHIM syndrome[1]. Uses: Scientific research. Group: Signaling pathways. Alternative Names: AMD-070 trihydrochloride; AMD-11070 trihydrochloride. CAS No. 2309699-17-8. Pack Sizes: 10 mM * 1 mL; 2 mg; 5 mg; 10 mg; 50 mg; 100 mg. Product ID: HY-50101A.
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