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Epalrestat Dimer Impurity. Uses: For analytical and research use. Group: Impurity standards. Molecular Formula: C30H26N2O6S4. Mole Weight: 638.79. Catalog: APB07847.
Epalrestat (E, E)-Isomer
A stereoisomer of Epalrestat. Epalrestat is a carboxylic acid-based inhibitor of aldose reductase. Synonyms: 2-((Z)-5-((Z)-2-Methyl-3-phenylallylidene)-4-oxo-2-thioxothiazolidin-3-yl)acetic acid. Grades: > 95%. Molecular formula: C15H13NO3S2. Mole weight: 319.40.
Epalrestat (E, E)-Isomer
Epalrestat (E, E)-Isomer. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: 2-((E)-5-((E)-2-methyl-3-phenylallylidene)-4-oxo-2-thioxothiazolidin-3-yl)acetic acid. CAS No. 863988-85-6. Molecular Formula: C15H13NO3S2. Mole Weight: 319.40. Catalog: APB863988856.
Epalrestat (E, Z)-Isomer
Epalrestat (E, Z)-Isomer. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: 2-((E)-5-((Z)-2-methyl-3-phenylallylidene)-4-oxo-2-thioxothiazolidin-3-yl)acetic acid. CAS No. 124782-64-5. Molecular Formula: C15H13NO3S2. Mole Weight: 319.40. Catalog: APB124782645.
Epalrestat (E, Z)-Isomer
A stereoisomer of Epalrestat. Epalrestat is a carboxylic acid-based inhibitor of aldose reductase. Synonyms: (E,Z)-5-(2-Methyl-3-phenyl-2-propen-1-ylidene)-4-oxo-2-thioxo-3-thiazolidineacetic Acid. Grades: > 95%. Molecular formula: C15H13NO3S2. Mole weight: 319.40.
Epalrestat Impurity 10
Epalrestat Impurity 10. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: (Z)-2-methyl-3-phenylacrylaldehyde. CAS No. 66051-14-7. Molecular Formula: C10H10O. Mole Weight: 146.19. Catalog: APB66051147.
Epalrestat Impurity 13
Epalrestat Impurity 13. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: ammonium 2-(sulfonatomethanethioamido)acetate. Molecular Formula: C3H3NO5S2·2NH4. Mole Weight: 233.27. Catalog: APB05552.
Epalrestat Impurity 14
Epalrestat Impurity 14. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: isopropyl 2-((Z)-5-((E)-2-methyl-3-phenylallylidene)-4-oxo-2-thioxothiazolidin-3-yl)acetate. Molecular Formula: C18H19NO3S2. Mole Weight: 361.48. Catalog: APB05551.
Epalrestat Impurity 15
Epalrestat Impurity 15. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: (E)-1-phenylhept-1-en-3-ol. CAS No. 109801-00-5. Molecular Formula: C13H18O. Mole Weight: 190.28. Catalog: APB109801005.
Epalrestat Impurity 16
Epalrestat Impurity 16. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: 76046-54-3 (free acid); ammonium 2, 2'- (disulfannebis (carbonothioyl)bis (azanediyl))diacetate. Molecular Formula: C6H6N2O4S4·2NH4. Mole Weight: 334.46. Catalog: APB05550.
Epalrestat Impurity 17
Epalrestat Impurity 17. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: 2041-59-0 (free acid); ammonium 2-(dithiocarboxylatoamino)acetate. Molecular Formula: C3H3NO2S2·2NH4. Mole Weight: 185.27. Catalog: APB05549.
Epalrestat Impurity 19
Epalrestat Impurity 19. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: 2-(2,4-dioxothiazolidin-3-yl)acetic acid. CAS No. 31061-24-2. Molecular Formula: C5H5NO4S. Mole Weight: 175.16. Catalog: APB31061242.
Epalrestat Impurity 20
Epalrestat Impurity 20. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: ethyl 2-(4-oxo-2-thioxothiazolidin-3-yl)acetate. CAS No. 23176-01-4. Molecular Formula: C7H9NO3S2. Mole Weight: 219.28. Catalog: APB23176014.
Epalrestat Impurity 21
Epalrestat Impurity 21. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: (E)-2-(4-oxo-5-propylidene-2-thioxothiazolidin-3-yl)acetic acid. Molecular Formula: C8H9NO3S2. Mole Weight: 231.29. Catalog: APB05548.
Epalrestat Impurity 22
Epalrestat Impurity 22. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: methyl 2-((Z)-5-((E)-2-methyl-3-phenylallylidene)-4-oxo-2-thioxothiazolidin-3-yl)acetate. Molecular Formula: C16H15NO3S2. Mole Weight: 333.43. Catalog: APB05547.
Epalrestat Impurity 23
Epalrestat Impurity 23. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: 2-((Z)-4-oxo-5-((E)-3-phenylallylidene)-2-thioxothiazolidin-3-yl)acetic acid. CAS No. 1800597-47-0. Molecular Formula: C14H11NO3S2. Mole Weight: 305.37. Catalog: APB1800597470.
Epalrestat Impurity 24
Epalrestat Impurity 24. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: (Z)-5-((E)-2-methyl-3-phenylallylidene)-2-thioxothiazolidin-4-one. CAS No. 15289-56-2. Molecular Formula: C13H11NOS2. Mole Weight: 261.36. Catalog: APB15289562.
Epalrestat Impurity 25
Epalrestat Impurity 25. Uses: For analytical and research use. Group: Impurity standards. Molecular Formula: C30H26N2O6S4. Mole Weight: 638.79. Catalog: APB07849.
Epalrestat Impurity 25
Epalrestat Impurity 25. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: (E)-2-methyl-3-phenylacrylaldehyde. CAS No. 15174-47-7. Molecular Formula: C10H10O. Mole Weight: 146.19. Catalog: APB15174477.
Epalrestat Impurity 26
Epalrestat Impurity 26. Uses: For analytical and research use. Group: Impurity standards. Molecular Formula: C16H15NO3S2. Mole Weight: 333.42. Catalog: APB07848.
Epalrestat Impurity 26
Epalrestat Impurity 26. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: 2-(5-oxo-2-thioxothiazolidin-3-yl)acetic acid. CAS No. 179027-75-9. Molecular Formula: C5H5NO3S2. Mole Weight: 190.97. Catalog: APB179027759.
Epalrestat Impurity 27
Epalrestat Impurity 27. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: 39680-96-1; 2-(dithiocarboxyamino)acetic acid,ammonium salt. CAS No. 6861-95-6. Molecular Formula: C3H11N3O2S2. Mole Weight: 185.27. Catalog: APB6861956.
Epalrestat Impurity 28
Epalrestat Impurity 28. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: 2-(4-oxo-2-thioxothiazolidin-3-yl)acetamide. CAS No. 39486-57-2. Molecular Formula: C5H6N2O2S2. Mole Weight: 190.24. Catalog: APB39486572.
Epalrestat Impurity 28
Epalrestat Impurity 28. Uses: For analytical and research use. Group: Impurity standards. CAS No. 98984-15-7. Molecular Formula: C8H9NO3S2. Mole Weight: 231.28. Catalog: APB98984157.
Epalrestat Impurity 29
Epalrestat Impurity 29. Uses: For analytical and research use. Group: Impurity standards. CAS No. 15250-29-0. Molecular Formula: C10H10O2. Mole Weight: 162.19. Catalog: APB15250290.
Epalrestat Impurity 29
Epalrestat Impurity 29. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: methyl 2-(4-oxo-2-thioxothiazolidin-3-yl)acetate. CAS No. 149789-77-5. Molecular Formula: C6H7NO3S2. Mole Weight: 205.25. Catalog: APB149789775.
Epalrestat Impurity 3
Epalrestat Impurity 3. Uses: For analytical and research use. Group: Impurity standards. CAS No. 682775-70-8. Molecular Formula: C16H15NO3S2. Mole Weight: 333.42. Catalog: APB682775708.
Epalrestat Impurity 30
Epalrestat Impurity 30. Uses: For analytical and research use. Group: Impurity standards. Molecular Formula: C11H12O. Mole Weight: 160.22. Catalog: APB07850.
Epalrestat Impurity 30
Epalrestat Impurity 30. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: 2-(5-benzylidene-4-oxo-2-thioxothiazolidin-3-yl)acetic acid. CAS No. 82159-06-6. Molecular Formula: C12H9NO3S2. Mole Weight: 279.33. Catalog: APB82159066.
Epalrestat Impurity 31
Epalrestat Impurity 31. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: 3-hydroxy-2-methyl-3-phenylpropanal. Molecular Formula: C10H12O2. Mole Weight: 164.20. Catalog: APB05907.
Epalrestat Impurity 32
Epalrestat Impurity 32. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: (Z)-3-methyl-4-phenylbut-3-enal. Molecular Formula: C11H12O. Mole Weight: 160.21. Catalog: APB05905.
Epalrestat Impurity 33
Epalrestat Impurity 33. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: (2-amino-2-oxoethyl)carbamodithioic acid. Molecular Formula: C3H6N2OS2. Mole Weight: 150.22. Catalog: APB05906.
Epalrestat Impurity 33 (Ammonium Salt)
Epalrestat Impurity 33 (Ammonium Salt). Uses: For analytical and research use. Group: Impurity standards. Alternative Names: (2-amino-2-oxoethyl)carbamodithioic acid,ammonium salt. Molecular Formula: C3H5N2OS2·NH4. Mole Weight: 167.25. Catalog: APB05903.
Epalrestat Impurity 34
Epalrestat Impurity 34. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: 2- ( ( (carboxymethyl) carbamothioyl) thio) acetic acid. CAS No. 29677-65-4. Molecular Formula: C5H7NO4S2. Mole Weight: 209.24. Catalog: APB29677654.
Epalrestat Impurity 35
Epalrestat Impurity 35. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: (E)-2-(5-benzylidene-4-oxo-2-thioxothiazolidin-3-yl)acetic acid. Molecular Formula: C12H9NO3S2. Mole Weight: 279.33. Catalog: APB05904.
Epalrestat Impurity 36
Epalrestat Impurity 36. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: 2-chloro-2-((Z)-5-((E)-2-methyl-3-phenylallylidene)-4-oxo-2-thioxothiazolidin-3-yl)acetic acid. Molecular Formula: C15H12ClNO3S2. Mole Weight: 353.84. Catalog: APB05902.
Epalrestat Impurity 37
Epalrestat Impurity 37. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: (Z)-2-methyl-3-phenylacrylic acid. Molecular Formula: C10H10O2. Mole Weight: 162.19. Catalog: APB05901.
Epalrestat Impurity 38
Epalrestat Impurity 38. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: 2-chloro-2-(4-oxo-2-thioxothiazolidin-3-yl)acetic acid. Molecular Formula: C5H4ClNO3S2. Mole Weight: 225.67. Catalog: APB05900.
Epalrestat Impurity 39
Epalrestat Impurity 39. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: (2-ethoxy-2-oxoethyl)carbamodithioic acid. CAS No. 44912-47-2. Molecular Formula: C5H9NO2S2. Mole Weight: 179.26. Catalog: APB44912472.
Epalrestat Impurity 40
Epalrestat Impurity 40. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: 2-(2-(dithiocarboxyamino)acetamido)acetic acid. CAS No. 138722-76-6. Molecular Formula: C5H8N2O3S2. Mole Weight: 208.26. Catalog: APB138722766.
Epalrestat Impurity 41
Epalrestat Impurity 41. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: ammonium (2-((2-((carboxymethyl)amino)-2-oxoethyl)amino)-2-oxoethyl)carbamodithioate. Molecular Formula: C7H14N4O4S2. Mole Weight: 282.34. Catalog: APB05899.
Epalrestat Impurity 42
Epalrestat Impurity 42. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: 2-(2-(4-oxo-2-thioxothiazolidin-3-yl)acetamido)acetic acid. CAS No. 190773-76-3. Molecular Formula: C7H8N2O4S2. Mole Weight: 248.28. Catalog: APB190773763.
Epalrestat Impurity 43
Epalrestat Impurity 43. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: 2-(2-(2-(4-oxo-2-thioxothiazolidin-3-yl)acetamido)acetamido)acetic acid. Molecular Formula: C9H11N3O5S2. Mole Weight: 305.33. Catalog: APB05897.
Epalrestat Impurity 44
Epalrestat Impurity 44. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: (E)-2-(3-(carboxymethyl)-4-oxo-2-thioxothiazolidin-5-ylidene)acetic acid. Molecular Formula: C7H5NO5S2. Mole Weight: 247.25. Catalog: APB05898.
Epalrestat Impurity 45
Epalrestat Impurity 45. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: 2,2-dichloro-N,N-dimethylacetamide. CAS No. 5468-76-8. Molecular Formula: C4H7Cl2NO. Mole Weight: 156.01. Catalog: APB5468768.
Epalrestat Impurity 46
Epalrestat Impurity 46. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: 2,2-dimethoxy-N,N-dimethylacetamide. CAS No. 25408-61-1. Molecular Formula: C6H13NO3. Mole Weight: 147.17. Catalog: APB25408611.
Epalrestat Impurity 47
Epalrestat Impurity 47. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: 2-((Z)-2,4-dioxo-5-((E)-3-phenylallylidene)thiazolidin-3-yl)acetic acid. Molecular Formula: C14H11NO4S. Mole Weight: 289.31. Catalog: APB05896.
Epalrestat Impurity 48
Epalrestat Impurity 48. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: 2-(5-chloro-4-oxo-2-thioxothiazolidin-3-yl)acetic acid. Molecular Formula: C5H4ClNO3S2. Mole Weight: 225.67. Catalog: APB05895.
Epalrestat Impurity 7
Epalrestat Impurity 7. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: (Z)-2-(4-oxo-5-propylidene-2-thioxothiazolidin-3-yl)acetic acid. CAS No. 130786-32-2. Molecular Formula: C8H9NO3S2. Mole Weight: 231.29. Catalog: APB130786322.
Epalrestat Impurity 8
Epalrestat Impurity 8. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: 2-(4-oxo-2-thioxothiazolidin-3-yl)acetic acid. CAS No. 5718-83-2. Molecular Formula: C5H5NO3S2. Mole Weight: 191.23. Catalog: APB5718832.
Epalrestat Impurity A
Epalrestat Impurity A. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: ethyl 2-((Z)-5-((E)-2-methyl-3-phenylallylidene)-4-oxo-2-thioxothiazolidin-3-yl)acetate. CAS No. 682775-71-9. Molecular Formula: C17H17NO3S2. Mole Weight: 347.45. Catalog: APB682775719.
Epalrestat Impurity E
Epalrestat Impurity E. Uses: For analytical and research use. Group: Impurity standards. Molecular Formula: C11H13NO3S2. Mole Weight: 271.35. Catalog: APB07846.
Epalrestat Oxide
Epalrestat Oxide. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: 2-((Z)-5-((E)-2-methyl-3-phenylallylidene)-2,4-dioxothiazolidin-3-yl)acetic acid. CAS No. 794510-29-5. Molecular Formula: C15H13NO4S. Mole Weight: 303.33. Catalog: APB794510295.
Epalrestat (Z, Z)-Isomer
A stereoisomer of Epalrestat. Epalrestat is a carboxylic acid-based inhibitor of aldose reductase. Synonyms: 2-((Z)-5-((Z)-2-Methyl-3-phenylallylidene)-4-oxo-2-thioxothiazolidin-3-yl)acetic acid. Grades: > 95%. Molecular formula: C15H13NO3S2. Mole weight: 319.40.
Epalrestat (Z, Z)-Isomer
Epalrestat (Z, Z)-Isomer. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: 2-((Z)-5-((Z)-2-methyl-3-phenylallylidene)-4-oxo-2-thioxothiazolidin-3-yl)acetic acid. CAS No. 124782-63-4. Molecular Formula: C15H13NO3S2. Mole Weight: 319.4. Catalog: APB124782634.
Epalrestat (Z, Z)-Isomer Methyl Ester
Epalrestat (Z, Z)-Isomer Methyl Ester. Uses: For analytical and research use. Group: Impurity standards. Alternative Names: methyl 2-((Z)-5-((Z)-2-methyl-3-phenylallylidene)-4-oxo-2-thioxothiazolidin-3-yl)acetate. Molecular Formula: C16H15NO3S2. Mole Weight: 333.43. Catalog: APB01890.
Epanorin
Epanorin is a lichen metabolite that can inhibit the proliferation of MCF-7 breast cancer cells. Synonyms: L-Leucine, N-[(3-hydroxy-5-oxo-4-phenyl-2(5H)-furanylidene)phenylacetyl]-, methyl ester; N-[2-(3-Hydroxy-5-oxo-4-phenyl-2(5H)-furanylidene)-2-phenylacetyl]-L-leucine methyl ester; (-)-Epanorin. CAS No. 18463-10-0. Molecular formula: C25H25NO6. Mole weight: 435.47.
EP Chlorpheniramine Maleate Impurity A (2HCl salt form)
An impurity of Chlorpheniramine. Chlorpheniramine is an antihistamine used to prevent symptoms of allergy. It acts via inhibiting histamine produced during anaphylaxis. Synonyms: 2-(4-Chlorophenyl)-4-(dimethylamino)-2-(2-(dimethylamino)ethyl)butanenitrile; 2-(4-Chlorophenyl)-4-(dimethylamino)-2-[2-(dimethylamino)ethyl]butanenitrile dihydrochloride. Grades: 95%. Molecular formula: C16H26Cl3N3. Mole weight: 366.761.
Epc-k(1)
Heterocyclic Organic Compound. Alternative Names: EPC-K(1);2-O-[[[(2R)-3,4-Dihydro-2,5,7,8-tetramethyl-2-[(4R,8R)-4,8,12-trimethyltridecyl]-2H-1-benzopyran]-6-yloxy](potassiooxy)phosphinyl]-L-ascorbic acid. CAS No. 127061-56-7. Catalog: ACM127061567.
Epcoritamab
Epcoritamab (GEN3013) is an bispecific IgG1 antibody redirecting T-cells toward CD3×CD20 + tumor cells. Epcoritamab induces potent T-cell-mediated cytotoxicity towards B-cell NHL cell lines [1]. Uses: Scientific research. Group: Inhibitory antibodies. Alternative Names: GEN3013. CAS No. 2134641-34-0. Pack Sizes: 1 mg; 5 mg; 10 mg. Product ID: HY-P99931.
EPDM
EPDM. Group: Polymers. CAS No. 25038-36-2.
EPDM chip
EPDM chip. Group: Polymers.
EPDM Rubber
EPDM Rubber. Group: Polymers.
Epelmycin A
It is produced by the strain of Streptomyces violaceus A262. It has anti-gram positive, negative bacteria and candida albicans activity, and has anti-leukemic L1210 activity, which is stronger than Aclacinomycin. Synonyms: 1-Naphthacenecarboxylic acid, 2-ethyl-1,2,3,4,6,11-hexahydro-2,5,7,12-tetrahydroxy-6,11-dioxo-4-((2,3,6-trideoxy-3-(dimethylamino)-4-O-((2S-(2alpha,5beta(2S*,6R*),6beta))-tetrahydro-6-methyl-5-((tetrahydro-6-methyl-5-oxo-2H-pyran-2-yl)oxy)-2H-pyran-2-yl)-alpha-L-lyxo-hexopyranosyl)oxy)-, methyl ester. CAS No. 107807-25-0. Molecular formula: C42H53NO15. Mole weight: 811.87.
Epelmycin B
It is produced by the strain of Streptomyces violaceus A262. It has anti-gram positive, negative bacteria and candida albicans activity, and has anti-leukemic L1210 activity, which is stronger than Aclacinomycin. Synonyms: 11-Hydroxyauramycin B. CAS No. 107807-24-9. Molecular formula: C42H51NO16. Mole weight: 825.85.
Epelmycin C
It is produced by the strain of Streptomyces violaceus A262. It has anti-gram positive, negative bacteria and candida albicans activity, and has anti-leukemic L1210 activity, which is stronger than Aclacinomycin. Synonyms: 1-Naphthacenecarboxylic acid, 2-ethyl-1,2,3,4,6,11-hexahydro-2,5,7,12-tetrahydroxy-6,11-dioxo-4-((2,3,6-trideoxy-4-O-(2,6-dideoxy-alpha-L-lyxo-hexopyranosyl)-3-(dimethylamino)-alpha-L-lyxo-hexopyranosyl)oxy)-, methyl ester. CAS No. 107807-23-8. Molecular formula: C36H45NO14. Mole weight: 715.74.
Epelmycin D
It is produced by the strain of Streptomyces violaceus A262. It has anti-gram positive, negative bacteria and candida albicans activity, and has anti-leukemic L1210 activity, which is stronger than Aclacinomycin. Synonyms: Violamycin A4; 1-Naphthacenecarboxylic acid, 2-ethyl-1,2,3,4,6,11-hexahydro-2,5,7,12-tetrahydroxy-6,11-dioxo-4-((2,3,6-trideoxy-3-(dimethylamino)-alpha-L-lyxo-hexopyranosyl)oxy)-, methyl ester. CAS No. 107807-22-7. Molecular formula: C30H35NO11. Mole weight: 585.60.
Epelmycin E
It is produced by the strain of Streptomyces violaceus A262. It has anti-gram positive, negative bacteria and candida albicans activity, and has anti-leukemic L1210 activity, which is stronger than Aclacinomycin. Synonyms: 11-Hydroxyaclacinomycin A; 1-Naphthacenecarboxylic acid,1,2,3,4,6,11-hexahydro-6,11-dioxo-2-ethyl-2,5,7,12-tetrahydroxy-4-((2,3,6-trideoxy-4-O-(2,6-dideoxy-4-O-((2R-trans)-tetrahydro-6-methyl-5-oxo-2H-pyran-2-yl)-alpha-L-lyxo-hexopyranosyl)-3-(dimethylamino)-alpha-L-lyxo-hexopyranosyl)oxy)-, methyl ester, (1R-(1-alpha,2-beta,4-beta))-; sigma-Rmn-A; epsilon-RMN-A. CAS No. 76264-93-2. Molecular formula: C42H53NO16. Mole weight: 827.87.
Epelsiban
Epelsiban is an oxytocin receptor antagonist under the developement of GlaxoSmithKline. It has high affinity for the oxytocin receptor (Ki = 0.13 nM) with >31,000-fold selectivity over the related vasopressin receptors. No development was reported about Phase II clinical tirals for the treatment of premature ejaculation. Uses: Premature ejaculation. Synonyms: GSK-557296; GSK 557296; GSK557296; GSK-557,296-B;(3R,6R)-6-((S)-sec-butyl)-3-(2,3-dihydro-1H-inden-2-yl)-1-((R)-1-(2,6-dimethylpyridin-3-yl)-2-morpholino-2-oxoethyl)piperazine-2,5-dione;1159097-48-9(besylate). Grades: 98%. CAS No. 872599-83-2. Molecular formula: C30H38N4O4. Mole weight: 518.65.
Epelsiban besylate
This active molecular, also known as GSK-557296B is a selective, sub-nanomolar (Ki=0.13 nM) oxytocin receptor antagonist with more than 30000-fold selectivity over the related vasopressin receptors. GlaxoSmithKline developed it for the treatment of premature ejaculation in men and also as an agent to enhance embryo or blastocyst implantation in women undergoing embryo or blastocyst transfer associated with in vitro fertilization. In Jul 1st 2016, Phase-II clinical trials in Adenomyosis in USA was on going. In Jun 13th 2016, GlaxoSmithKline terminated phase I trial in Infertility (In volunteers) in USA. Uses: Adenomyosis;infertility; premature ejaculation. Synonyms: (3R,6R)-3-(2,3-Dihydro-1H-inden-2-yl)-1-((1R)-1-(2,6-dimethylpyridin-3-yl)-2- (morpholin-4-yl)-2-oxoethyl)-6-((1S)-1-methylpropyl)piperazine-2,5-dione monobenzenesulfonate,UNII-H629P9T4UN; UNII-H629P9T4UN; GSK557296B; GSK-557296B; 872599-83-2(free base). Grades: 98%. CAS No. 1159097-48-9. Molecular formula: C36H44N4O7S. Mole weight: 676.83.